| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| ALK |
HGNC:427 |
Q9UM73 |
1-[4-(2-ethoxy-2-oxoethyl)-2,3-dioxo-7-(trifluoromethyl)-1H-quinoxalin-6-yl]pyrrole-3-carboxylic acid |
15337998 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
n'-(4-Ethoxycarbonylphenyl)-n-(1-(6-trifluoromethyl-quinoxaline-2,3(1h,4h)dion-7-yl)pyrrol-3-ylmethyl)urea |
15840183 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
N'-(4-Carboxyphenyl)-N-(1-(6-trifluoromethylquinoxaline-2,3-(1H,4H) dion-7-yl)pyrrol-3-ylmethyl)urea |
15840184 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
(R)-5-(6-((4-methylpiperazin-1-yl)methyl)-1H-benzo[d]imidazol-1-yl)-3-(1-(2-(trifluoromethyl)phenyl)ethoxy)thiophene-2-carboxamide |
15983966 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
Azd-1152hqpa |
16007391 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
5-chloro-N4-(2-(isopropylsulfonyl)phenyl)-N2-(2-methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)phenyl)pyrimidine-2,4-diamine |
16038120 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
Gsk-690693 |
16725726 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
Pictilisib |
17755052 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
N-(3-(5-chloro-1H-pyrrolo[2,3-b]pyridine-3-carbonyl)-2,4-difluorophenyl)propane-1-sulfonamide |
24180719 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
[6-chloro-4-methyl-3-[[3-(methylsulfamoylamino)phenyl]methyl]-2-oxochromen-7-yl] N,N-dimethylcarbamate |
24753787 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
Isobutyl4-(7-amino-3-(4-(4-methylpiperazin-1-yl)phenyl)pyrazolo[1,5-a]pyrimidin-6-yl)phenylcarbamate |
24762205 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
5-(2-aminopyrimidin-4-yl)-2-phenyl-1H-pyrrole-3-carboxamide |
24809764 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
1-methyl-8-(5-(4-methylpiperazin-1-yl)-2-(trifluoromethoxy)phenylamino)-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide |
24825755 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
(S)-1-benzyl-7-(4-(2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl)phenyl)-3,4-dihydropyrido[2,3-b]pyrazin-2(1H)-one |
24852349 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
Quizartinib |
24889392 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
4-(2-Chloro-4-fluorophenyl)-8-(2,6-dichlorophenyl)-7-oxido-1,7-naphthyridin-7-ium |
24896769 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
1H-Pyrazolo[4,3-h]quinazoline-3-carboxamide, 4,5-dihydro-8-[[2-methoxy-5-(4-methyl-1-piperazinyl)phenyl]amino]-1-methyl- |
24993189 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
2-[5-Chloro-2-(1-methyl-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-ylamino)-pyrimidin-4-ylamino]-N-methyl-benzenesulfonamide |
25157614 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
N-[5-(3,5-Difluorobenzyl)-1h-Indazol-3-Yl]-2-[(4-Hydroxycyclohexyl)amino]-4-(4-Methylpiperazin-1-Yl) Benzamide |
25176165 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
2-((2-((1-(2-(Dimethylamino)acetyl)-5-methoxyindolin-6-yl)amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino)-6-fluoro-N-methylbenzamide |
25182616 |
BindingDB |