| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| ALK |
HGNC:427 |
Q9UM73 |
5-Benzo[1,3]dioxol-5-ylmethyl-10-fluoro-8-(4-methyl-piperazin-1-yl)-[1,2,4]triazolo[1,5-c]quinazolin-2-ylamine |
51037948 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
(S)-3-Hydroxy Midostaurin |
52945601 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
Infigratinib |
53235510 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
2-(7-(5-chloro-4-(2-methoxy-4-morpholinophenylamino)pyrimidin-2-ylamino)-8-methoxy-4,5-dihydro-1H-benzo[d]azepin-3(2H)-yl)-N-methylacetamide |
53317655 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
5-chloro-N2-(8-methoxy-3-(2-(methylsulfonyl)ethyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)-N4-(2-methoxy-4-morpholinophenyl)pyrimidine-2,4-diamine |
53318636 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
(3S,5Z,9S)a9,16aDihydroxya14amethoxya3amethyla3,4,7,8,9,10,11,12aoctahydroa1Ha2abenzoxacyclotetradecinea1,7adione |
53324451 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
6,6-Dimethyl-8-(1-oxetan-3-yl-piperidin-4-yl)-11-oxo-6,11-dihydro-5H-benzo[b]carbazole-3-carbonitrile |
53357328 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
1-[5-Tert-Butyl-3-({4-[2-(Dimethylamino)ethyl]-5-Oxo-1,4-Diazepan-1-Yl}carbonyl)thiophen-2-Yl]-3-(2,3-Dichlorophenyl)urea |
53384644 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
N-[2-[2-[4-[4-[(2S)-2-hydroxypropyl]piperazin-1-yl]-2-methoxyanilino]pyrrolo[2,1-f][1,2,4]triazin-7-yl]phenyl]-N-methylmethanesulfonamide |
53465297 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
[2-Methoxy-4-(4-methyl-piperazin-1-yl)-phenyl]-[7-(2-methoxy-phenyl)-pyrrolo[2,1-f][1,2,4]triazin-2-yl]-amine |
54577897 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
(2S)-1-[4-[3-methoxy-4-[[7-(2-methoxyphenyl)pyrrolo[2,1-f][1,2,4]triazin-2-yl]amino]phenyl]piperazin-1-yl]propan-2-ol |
54578104 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
3-bromo-8-(2-(diethylamino)ethoxy)-6,6-dimethyl-5H-benzo[b]carbazol-11(6H)-one |
54587776 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
(3S)-N-[[4-(trifluoromethoxy)phenyl]methyl]-1-[2-(3,4,5-trimethoxyanilino)pyrimidin-4-yl]piperidine-3-carboxamide |
54596950 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
Spiro[piperidine-4,3'-[3H]pyrido[3,4-b]indole]-4'-carbonitrile, 7',8'-dichloro-1',2',4',9'-tetrahydro-9'-methyl-1'-oxo- |
54613583 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
Azd3463 |
56599293 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
N-[6-[[4-(2-hydroxypropan-2-yl)piperidin-1-yl]methyl]-1-[4-(propan-2-ylcarbamoyl)cyclohexyl]benzimidazol-2-yl]pyridine-4-carboxamide |
56650031 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
3-cyano-N-[6-[[4-(2-hydroxypropan-2-yl)piperidin-1-yl]methyl]-1-[4-(propan-2-ylcarbamoyl)cyclohexyl]benzimidazol-2-yl]benzamide |
56650355 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
4-fluoro-N-[6-[[(2-hydroxy-2-methylpropyl)amino]methyl]-1-[4-(propan-2-ylcarbamoyl)cyclohexyl]benzimidazol-2-yl]benzamide |
56650694 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
Ethyl 4-[2-benzamido-6-(piperidin-1-ylmethyl)benzimidazol-1-yl]cyclohexane-1-carboxylate |
56653076 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
4-fluoro-N-[6-[[3-(2-hydroxypropan-2-yl)azetidin-1-yl]methyl]-1-[4-(propan-2-ylcarbamoyl)cyclohexyl]benzimidazol-2-yl]benzamide |
56654815 |
BindingDB |