| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| ALK |
HGNC:427 |
Q9UM73 |
6-(6-Fluoroindol-1-yl)-2-[2-[7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxyethyl]pyridazin-3-one |
73386831 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
2-[(1r)-1-{[3-Amino-6-(2-Methoxypyridin-3-Yl)pyrazin-2-Yl]oxy}ethyl]-4-Fluoro-N-Methylbenzamide |
73819542 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
3-[(1R)-1-[5-fluoro-2-(triazol-2-yl)phenyl]ethoxy]-5-(3-methylsulfonylphenyl)pyridin-2-amine |
73819543 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
(10r)-7-Amino-3-Cyclopropyl-12-Fluoro-1,10,16-Trimethyl-16,17-Dihydro-1h-8,4-(Metheno)pyrazolo[4,3-H][2,5,11]benzoxadiazacyclotetradecin-15(10h)-One |
73819548 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
N-[5-[(3,5-difluorophenyl)methyl]-2,3,3a,4,5,6,7,7a-octahydro-1H-indazol-3-yl]-4-(4-methylpiperazin-1-yl)-2-(oxan-4-ylamino)benzamide |
74394320 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
2-[[2-[(3,5-dimethyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)amino]pyrido[3,2-d]pyrimidin-4-yl]amino]-N-methylbenzamide |
76282402 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
5-(1,3-dimethylpyrazol-4-yl)-3-[(1R)-1-[5-fluoro-2-(triazol-2-yl)phenyl]ethoxy]pyridin-2-amine |
76311144 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
7-Bromo-4-chloropyrazino[1,2-a]benzimidazole |
76317830 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
N-(3-nitrophenyl)pyrimido[1,6-a]benzimidazol-3-amine |
76321540 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
4-Chloropyrazino[1,2-a]benzimidazole |
76321541 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
3-Chloropyrimido[1,6-a]benzimidazole |
76325144 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
8-Bromo-3-(4-methoxyphenyl)pyrimido[1,6-a]benzimidazole |
76328703 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
8-Bromo-3-chloropyrimido[1,6-a]benzimidazole |
76332386 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
4,7-Bis[4-(4-methylpiperazin-1-yl)phenyl]pyrazino[1,2-a]benzimidazole |
76332387 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
Envonalkib |
76899983 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
Lorlatinib (PF-06463922) |
78162481 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
5-chloro-2-N-(7-methoxy-1,2,3,4-tetrahydroisoquinolin-6-yl)-4-N-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamine |
78319165 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
4-((1-(4-chloro-3-fluorobenzyl)-1H-pyrazol-5-yl)ethynyl)-5-(2-methoxy-4-(4-methylpiperazin-1-yl)phenyl)pyridin-2-amine |
78324677 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
3-[(3-Fluorophenoxy)methyl]-5-(1-piperidin-4-ylpyrazol-4-yl)pyridin-2-amine |
78324681 |
BindingDB |
| ALK |
HGNC:427 |
Q9UM73 |
Dalmelitinib |
86302574 |
BindingDB |