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Drugs And Genes
DRUGs and GENEs
GENE_SYMBOL HGNC_ID UNIPROT_ID DRUG_NAME PUBCHEM_CID Datasource
ADORA2A HGNC:263 P29274 3-cyano-N-cyclopropyl-5-[3-[5-[(3,5-dichloropyridin-4-yl)carbamoylamino]-1-ethyl-6-oxopyridazin-3-yl]phenyl]benzamide 67548983 BindingDB
ADORA2A HGNC:263 P29274 3-N-cyclopropyl-5-[3-[5-[(3,5-dichloropyridin-4-yl)carbamoylamino]-1-ethyl-6-oxopyridazin-3-yl]phenyl]-1-N-(2-morpholin-4-ylethyl)benzene-1,3-dicarboxamide 67549056 BindingDB
ADORA2A HGNC:263 P29274 1-N,3-N-dicyclopropyl-5-[3-[5-[(3,5-dichloropyridin-4-yl)carbamoylamino]-1-ethyl-6-oxopyridazin-3-yl]phenyl]benzene-1,3-dicarboxamide 67549097 BindingDB
ADORA2A HGNC:263 P29274 N-cyclopropyl-3-[3-[5-[(3,5-dichloropyridin-4-yl)carbamoylamino]-1-ethyl-6-oxopyridazin-3-yl]phenyl]-5-ethoxybenzamide 67549451 BindingDB
ADORA2A HGNC:263 P29274 3-N-(1-benzylpiperidin-4-yl)-1-N-cyclopropyl-5-[3-[5-[(3,5-dichloropyridin-4-yl)carbamoylamino]-1-ethyl-6-oxopyridazin-3-yl]phenyl]benzene-1,3-dicarboxamide 67549626 BindingDB
ADORA2A HGNC:263 P29274 3-N-cyclopropyl-5-[3-[5-[(3,5-dichloropyridin-4-yl)carbamoylamino]-1-ethyl-6-oxopyridazin-3-yl]phenyl]-1-N-(2-piperidin-1-ylethyl)benzene-1,3-dicarboxamide 67549879 BindingDB
ADORA2A HGNC:263 P29274 2-[6-amino-9-[(2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]purin-2-yl]sulfanylacetic acid 68148396 BindingDB
ADORA2A HGNC:263 P29274 4-[7-Amino-10-[2-[4-[4-(carboxymethoxy)phenyl]piperazin-1-yl]ethyl]-3,5,6,8,10,11-hexazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7,11-pentaen-4-yl]-4-hydroxybutanoic acid 68388533 BindingDB
ADORA2A HGNC:263 P29274 2-[4-[4-[2-[7-Amino-4-(furan-2-yl)-3,5,6,8,10,11-hexazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7,11-pentaen-10-yl]ethyl]piperazin-1-yl]phenoxy]acetic acid 68388551 BindingDB
ADORA2A HGNC:263 P29274 2-[7-Amino-4-(furan-2-yl)-3,5,6,8,10,11-hexazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7,11-pentaen-10-yl]acetic acid 68388674 BindingDB
ADORA2A HGNC:263 P29274 Methyl 3-[3-[5-[(3,5-dichloropyridin-4-yl)carbamoylamino]-1-ethyl-6-oxopyridazin-3-yl]phenyl]-5-[3-(dimethylamino)propylcarbamoyl]benzoate 68405754 BindingDB
ADORA2A HGNC:263 P29274 3-(cyclopropylmethoxy)-5-[3-[5-[(3,5-dichloropyridin-4-yl)carbamoylamino]-1-ethyl-6-oxopyridazin-3-yl]phenyl]-N-(2-piperidin-1-ylethyl)benzamide 68405874 BindingDB
ADORA2A HGNC:263 P29274 5-[3-[5-[(3,5-dichloropyridin-4-yl)carbamoylamino]-1-ethyl-6-oxopyridazin-3-yl]phenyl]-3-N-(2-hydroxyethyl)-1-N-(2-piperidin-1-ylethyl)benzene-1,3-dicarboxamide 68405927 BindingDB
ADORA2A HGNC:263 P29274 N-(2-hydroxyethyl)-2-imino-8-methoxychromene-3-carboxamide 70694477 BindingDB
ADORA2A HGNC:263 P29274 4-[2-[6-amino-9-[(2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]purin-2-yl]sulfonylethyl]benzenesulfonic acid 70694510 BindingDB
ADORA2A HGNC:263 P29274 N-(5-hydroxypentyl)-2-imino-8-methoxychromene-3-carboxamide 70696537 BindingDB
ADORA2A HGNC:263 P29274 trans-4-({1-[5-(5-fluoro-1H-benzimidazol-2-yl)pyridin-2-yl]piperidin-4-yl}oxy)cyclohexanecarboxylic acid 71078482 BindingDB
ADORA2A HGNC:263 P29274 2-[4-[1-[5-(1H-benzimidazol-2-yl)pyridin-2-yl]piperidin-4-yl]oxycyclohexyl]acetic acid 71110518 BindingDB
ADORA2A HGNC:263 P29274 2-Chloro-3'-deoxy-3'-fluoro-N-[(3-iodophenyl)methyl]adenosine 71364275 BindingDB
ADORA2A HGNC:263 P29274 (1S,2S,3R,4R,5S)-1-(6-aminopurin-9-yl)-4-(hydroxymethyl)bicyclo[3.1.0]hexane-2,3-diol 71450842 BindingDB