| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TIE1 |
HGNC:11809 |
P35590 |
2,6-Dimethylphenyl (2,4-dimethoxyphenyl)(2-((4-(4-methylpiperazin-1-yl)phenyl)amino)pyrimidin-4-yl)carbamate |
11844351 |
DSigDB |
| TIE1 |
HGNC:11809 |
P35590 |
R406 Benzenesulfonate |
11984591 |
DSigDB |
| TIE1 |
HGNC:11809 |
P35590 |
(R)-5-(6-((4-methylpiperazin-1-yl)methyl)-1H-benzo[d]imidazol-1-yl)-3-(1-(2-(trifluoromethyl)phenyl)ethoxy)thiophene-2-carboxamide |
15983966 |
Pubchem |
| TIE1 |
HGNC:11809 |
P35590 |
Azd-1152hqpa |
16007391 |
ChemBL, Pubchem |
| TIE1 |
HGNC:11809 |
P35590 |
5-chloro-N4-(2-(isopropylsulfonyl)phenyl)-N2-(2-methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)phenyl)pyrimidine-2,4-diamine |
16038120 |
DSigDB |
| TIE1 |
HGNC:11809 |
P35590 |
Fedratinib |
16722836 |
Pubchem |
| TIE1 |
HGNC:11809 |
P35590 |
Quizartinib |
24889392 |
Pubchem |
| TIE1 |
HGNC:11809 |
P35590 |
N-methyl-6-[[4-(2-propan-2-ylsulfonylanilino)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino]-3-pyridinecarboxamide |
25226483 |
DSigDB |
| TIE1 |
HGNC:11809 |
P35590 |
Foretinib |
42642645 |
Pubchem |
| TIE1 |
HGNC:11809 |
P35590 |
3-(4-amino-7-cyclopentyl-7H-pyrrolo[2,3-d]pyrimidin-5-yl)phenol |
44381237 |
ChemBL |
| TIE1 |
HGNC:11809 |
P35590 |
Dabrafenib |
44462760 |
DSigDB |
| TIE1 |
HGNC:11809 |
P35590 |
Merestinib |
44603533 |
GtoPDB |
| TIE1 |
HGNC:11809 |
P35590 |
3-[4-Amino-7-[3-(hydroxymethyl)cyclobutyl]pyrrolo[2,3-d]pyrimidin-5-yl]phenol |
49825075 |
ChemBL |
| TIE1 |
HGNC:11809 |
P35590 |
Azd-4547 |
51039095 |
DSigDB |
| TIE1 |
HGNC:11809 |
P35590 |
(E)-N-(4-((4-Ethylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-(2-(4-methoxy-1H-pyrrolo[2,3-b]pyridin-5-yl)vinyl)-4-methylbenzamide |
53302361 |
DSigDB |
| TIE1 |
HGNC:11809 |
P35590 |
N-[(3R)-8-[[5-chloro-4-[2-fluoro-6-(methylcarbamoyl)anilino]pyrimidin-2-yl]amino]-5,5-dimethyl-2-oxo-3,4-dihydro-1H-1-benzazepin-3-yl]pyrrolidine-1-carboxamide |
56597775 |
GtoPDB |
| TIE1 |
HGNC:11809 |
P35590 |
5-Chloro-4-(1H-indol-3-yl)-N-(2-methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)phenyl)pyrimidin-2-amine |
56655374 |
DSigDB |
| TIE1 |
HGNC:11809 |
P35590 |
[3-Cyano-5-[[[2,4-dimethyl-5-[6-(3-pyridinyl)-1H-imidazo[1,2-b]pyrazol-1-yl]phenyl]amino]carbonyl]phenyl]pentafluorosulfur |
71623052 |
ChemBL |
| TIE1 |
HGNC:11809 |
P35590 |
3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-[4-(diethylamino)butylamino]-1-methyl-4H-pyrimido[4,5-d]pyrimidin-2-one |
73265276 |
DSigDB |
| TIE1 |
HGNC:11809 |
P35590 |
[2-methyl-5-[[3-(trifluoromethyl)phenyl]carbamoyl]phenyl] N-(2,4-dimethoxyphenyl)-N-[2-[4-(4-methylpiperazin-1-yl)anilino]pyrimidin-4-yl]carbamate |
73707529 |
DSigDB |