| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TNK2 |
HGNC:19297 |
Q07912 |
MK-5108 |
24748204 |
ChemBL, Pubchem |
| TNK2 |
HGNC:19297 |
Q07912 |
Alisertib |
24771867 |
DGidb |
| TNK2 |
HGNC:19297 |
Q07912 |
Ponatinib |
24826799 |
DSigDB |
| TNK2 |
HGNC:19297 |
Q07912 |
Adavosertib |
24856436 |
DGidb |
| TNK2 |
HGNC:19297 |
Q07912 |
Ruxolitinib |
25126798 |
ChemBL, Pubchem |
| TNK2 |
HGNC:19297 |
Q07912 |
Asp-3026 |
25134326 |
ChemBL, Pubchem |
| TNK2 |
HGNC:19297 |
Q07912 |
Entrectinib |
25141092 |
ChemBL, DGidb, DrugBank, Pubchem, TTD |
| TNK2 |
HGNC:19297 |
Q07912 |
N3-(2,6-dimethylphenyl)-1-(3-methoxy-3-methylbutyl)-N6-(4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-1H-pyrazolo[3,4-d]pyrimidine-3,6-diamine |
25154877 |
TTD |
| TNK2 |
HGNC:19297 |
Q07912 |
(R)-4-(3-(2,6-dichlorophenylamino)-6-(phenylamino)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)butane-1,2-diol |
25154878 |
TTD |
| TNK2 |
HGNC:19297 |
Q07912 |
1-(4-(4-(2-(Isopropylsulfonyl)phenylamino)-1H-pyrrolo[2,3-b]pyridin-6-ylamino)-3-methoxyphenyl)piperidin-4-ol |
25195352 |
ChemBL |
| TNK2 |
HGNC:19297 |
Q07912 |
1-[4-[[4-Amino-5-chloro-6-(2-propan-2-ylsulfonylanilino)-2-pyrimidinyl]amino]-3-methoxyphenyl]-4-piperidinecarboxamide |
25226117 |
DSigDB |
| TNK2 |
HGNC:19297 |
Q07912 |
N-methyl-6-[[4-(2-propan-2-ylsulfonylanilino)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino]-3-pyridinecarboxamide |
25226483 |
DSigDB |
| TNK2 |
HGNC:19297 |
Q07912 |
N3-(2,6-dimethylphenyl)-N6-(3-fluoro-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-1-(3-methoxy-3-methylbutyl)-1H-pyrazolo[3,4-d]pyrimidine-3,6-diamine |
25263033 |
ChemBL, TTD |
| TNK2 |
HGNC:19297 |
Q07912 |
Vemurafenib |
42611257 |
ChemBL, DSigDB, Pubchem |
| TNK2 |
HGNC:19297 |
Q07912 |
Foretinib |
42642645 |
Pubchem |
| TNK2 |
HGNC:19297 |
Q07912 |
N-{4-[(6-Oxo-5,6-Dihydrobenzo[c][1,8]naphthyridin-1-Yl)amino]phenyl}benzamide |
44189332 |
ChemBL, TTD |
| TNK2 |
HGNC:19297 |
Q07912 |
(R)-5,6-diphenyl-N-((tetrahydrofuran-2-yl)methyl)furo[2,3-d]pyrimidin-4-amine |
44438314 |
TTD |
| TNK2 |
HGNC:19297 |
Q07912 |
(S)-6-(4-(2-(dimethylamino)ethoxy)phenyl)-5-phenyl-N-((tetrahydrofuran-2-yl)methyl)furo[2,3-d]pyrimidin-4-amine |
44438318 |
ChemBL, TTD |
| TNK2 |
HGNC:19297 |
Q07912 |
(S)-6-(4-((4-methylpiperazin-1-yl)methyl)phenyl)-5-phenyl-N-((tetrahydrofuran-2-yl)methyl)furo[2,3-d]pyrimidin-4-amine |
44438320 |
TTD |
| TNK2 |
HGNC:19297 |
Q07912 |
3-Cyclobutyl-1-(4-phenoxyphenyl)imidazo[1,5-a]pyrazin-8-amine |
44438839 |
ChemBL, TTD |