| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TNKS2 |
HGNC:15677 |
Q9H2K2 |
6,7-difluoro-3-[4-(2-hydroxypropan-2-yl)phenyl]-2H-pyrrolo[1,2-a]pyrazin-1-one |
71765180 |
ChemBL |
| TNKS2 |
HGNC:15677 |
Q9H2K2 |
6-fluoro-3-[4-(2-hydroxypropan-2-yl)phenyl]-2H-pyrrolo[1,2-a]pyrazin-1-one |
71765181 |
ChemBL |
| TNKS2 |
HGNC:15677 |
Q9H2K2 |
3-(4-(2-Hydroxypropan-2-yl)phenyl)-6-methylpyrrolo[1,2-a]pyrazin-1(2H)-one |
71765184 |
ChemBL |
| TNKS2 |
HGNC:15677 |
Q9H2K2 |
3-[4-(2-hydroxypropan-2-yl)phenyl]-2H-pyrrolo[1,2-a]pyrazin-1-one |
71765501 |
ChemBL |
| TNKS2 |
HGNC:15677 |
Q9H2K2 |
6-[4-(2-hydroxypropan-2-yl)phenyl]-2-methyl-5H-pyrazolo[1,5-a]pyrazin-4-one |
71765581 |
ChemBL |
| TNKS2 |
HGNC:15677 |
Q9H2K2 |
Tankyrase-IN-5 |
71765621 |
ChemBL |
| TNKS2 |
HGNC:15677 |
Q9H2K2 |
2-(4-(Trifluoromethyl)phenyl)-4A,5,7,7A-tetrahydrothieno[3,4-D]pyrimidin-4(3H)-one |
71819164 |
ChemBL, TTD |
| TNKS2 |
HGNC:15677 |
Q9H2K2 |
(4s)-3-{4-[6-Amino-5-(Pyrimidin-2-Yl)pyridin-3-Yl]phenyl}-5,5-Dimethyl-4-Phenyl-1,3-Oxazolidin-2-One |
72193935 |
ChemBL, TTD |
| TNKS2 |
HGNC:15677 |
Q9H2K2 |
Cyclohexanecarboxylic acid, 4-[[1-[[2-cyano-3-(trifluoromethyl)phenyl]methyl]-1,4-dihydro-2,4-dioxo-3(2H)-quinazolinyl]methyl]-, trans- |
72549316 |
ChemBL, TTD |
| TNKS2 |
HGNC:15677 |
Q9H2K2 |
4-[[5-Chloro-1-[[2-cyano-3-(trifluoromethyl)phenyl]methyl]-2,4-dioxoquinazolin-3-yl]methyl]cyclohexane-1-carboxylic acid |
72549539 |
ChemBL |
| TNKS2 |
HGNC:15677 |
Q9H2K2 |
4-[[1-[[2-Cyano-3-(trifluoromethyl)phenyl]methyl]-5-fluoro-2,4-dioxoquinazolin-3-yl]methyl]cyclohexane-1-carboxylic acid |
72549540 |
ChemBL |
| TNKS2 |
HGNC:15677 |
Q9H2K2 |
Tnks1/2-IN-1 |
72549541 |
ChemBL, TTD |
| TNKS2 |
HGNC:15677 |
Q9H2K2 |
4-[[1-[[2-Cyano-3-(trifluoromethyl)phenyl]methyl]-5,6-dimethyl-2,4-dioxoquinazolin-3-yl]methyl]cyclohexane-1-carboxylic acid |
72549542 |
ChemBL |
| TNKS2 |
HGNC:15677 |
Q9H2K2 |
4-[[1-[[2-Cyano-3-(trifluoromethyl)phenyl]methyl]-5-methoxy-2,4-dioxoquinazolin-3-yl]methyl]cyclohexane-1-carboxylic acid |
72549543 |
ChemBL |
| TNKS2 |
HGNC:15677 |
Q9H2K2 |
Cyclohexanecarboxylic acid, 4-[[1-[[2-cyano-3-(trifluoromethyl)phenyl]methyl]-1,4-dihydro-5-methyl-2,4-dioxo-3(2H)-quinazolinyl]methyl]-, trans- |
72549782 |
ChemBL, GtoPDB, TTD |
| TNKS2 |
HGNC:15677 |
Q9H2K2 |
2-(2-Hydroxy-1,1-dimethyl-ethyl)-5-methyl-1,2,4,10-tetrahydro-3-oxa-10-aza-phenanthren-9-one |
72699516 |
TTD |
| TNKS2 |
HGNC:15677 |
Q9H2K2 |
10-Methyl-3-propan-2-yl-1,3,4,5-tetrahydropyrano[4,3-c]isoquinolin-6-one |
72699517 |
TTD |
| TNKS2 |
HGNC:15677 |
Q9H2K2 |
8-Propan-2-yl-6,7,8,10-tetrahydropyrano[4,3-h][1,6]naphthyridin-5-one |
72699596 |
ChemBL, TTD |
| TNKS2 |
HGNC:15677 |
Q9H2K2 |
2-Tert-butyl-1,2,4,10-tetrahydro-3-oxa-10-aza-phenanthren-9-one |
72699600 |
TTD |
| TNKS2 |
HGNC:15677 |
Q9H2K2 |
3-Propan-2-yl-1,3,4,5-tetrahydropyrano[4,3-c]isoquinolin-6-one |
72699677 |
TTD |