| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-(4-Cyclopropyl-2,3-dihydro-1H-inden-1-yl)-3-(1H-indazol-4-yl)urea |
24777770 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-(5-Cyclopropyl-2,3-dihydro-1H-inden-1-yl)-3-(1H-indazol-4-yl)urea |
24777771 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-(4-tert-butyl-2,3-dihydro-1H-inden-1-yl)-3-(1H-indazol-4-yl)urea |
24777772 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-(1H-Indazol-4-yl)-3-(4-morpholin-1-yl-indan-1-yl)-urea |
24777773 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-(6,7-dihydro-5H-cyclopenta[b]pyridin-5-yl)-3-(1H-indazol-4-yl)urea |
24777889 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
2-[2-piperidin-1-yl-4-[4-(trifluoromethyl)anilino]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]-N-propan-2-ylpyridine-3-sulfonamide |
24782137 |
ChemBL |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
7-(3-ethylsulfonylpyridin-2-yl)-N-[4-(trifluoromethyl)phenyl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine |
24782138 |
ChemBL |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
2-cyclohexyloxy-7-[3-(trifluoromethyl)pyridin-2-yl]-N-[4-(trifluoromethylsulfonyl)phenyl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine |
24782139 |
ChemBL |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
2-(1-propan-2-ylpyrrolidin-3-yl)oxy-N-[4-(trifluoromethyl)phenyl]-7-[3-(trifluoromethyl)pyridin-2-yl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine |
24782140 |
ChemBL |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
2-(1-cyclohexylethoxy)-N-(1-methyl-3,4-dihydro-2H-quinolin-7-yl)-7-[3-(trifluoromethyl)pyridin-2-yl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine |
24782393 |
ChemBL |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
2-(1-cyclohexylethoxy)-7-[3-(trifluoromethyl)pyridin-2-yl]-N-[4-(trifluoromethylsulfonyl)phenyl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine |
24782394 |
ChemBL |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
2-cyclopentyloxy-7-[3-(trifluoromethyl)pyridin-2-yl]-N-[4-(trifluoromethylsulfonyl)phenyl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine |
24782395 |
ChemBL |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
2-(1-cyclohexylethoxy)-N-(4-pyrrolidin-1-ylsulfonylphenyl)-7-[3-(trifluoromethyl)pyridin-2-yl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine |
24782396 |
ChemBL |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
2-(1-cyclopropylethoxy)-N-(1-methyl-3,4-dihydro-2H-quinolin-7-yl)-7-[3-(trifluoromethyl)pyridin-2-yl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine |
24782639 |
ChemBL |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
2-(oxan-4-yloxy)-7-[3-(trifluoromethyl)pyridin-2-yl]-N-[4-(trifluoromethylsulfonyl)phenyl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine |
24782640 |
ChemBL |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
2-cyclopentyloxy-N-(1-methyl-3,4-dihydro-2H-quinolin-7-yl)-7-[3-(trifluoromethyl)pyridin-2-yl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine |
24782641 |
ChemBL |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
2-cyclohexyloxy-N-[2-methyl-4-(trifluoromethyl)phenyl]-7-[3-(trifluoromethyl)pyridin-2-yl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine |
24782642 |
ChemBL |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
2-cyclohexyloxy-N-(1-methyl-3,4-dihydro-2H-quinolin-7-yl)-7-[3-(trifluoromethyl)pyridin-2-yl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine |
24782643 |
ChemBL |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
(4-tert-Butyl-phenyl)-[7-(3-trifluoromethyl-pyridin-2-yl)-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl]-amine |
24782891 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
N-(4-(trifluoromethyl)phenyl)-7-(3-(trifluoromethyl)pyridin-2-yl)-6,7,8,9-tetrahydro-5H-pyrimido[5,4-d]azepin-4-amine |
24782892 |
ChemBL, TTD |