| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-[[2-(3-chlorophenyl)-5-(trifluoromethyl)pyrazol-3-yl]methyl]-3-(1H-indazol-4-yl)urea |
49803625 |
ChemBL |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-[[2-(3-Chlorophenyl)-5-(trifluoromethyl)pyrazol-3-yl]methyl]-3-(1-methylindazol-4-yl)urea |
49803911 |
ChemBL |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
N-[(5-tert-butyl-2-hexylpyrazol-3-yl)methyl]-2-[3-fluoro-4-(methanesulfonamido)phenyl]propanamide |
49804209 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
N-[[2-(3-chlorophenyl)-5-(trifluoromethyl)pyrazol-3-yl]methyl]-2-(3-fluorophenyl)-2-methylpropanamide |
49804215 |
ChemBL |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
N-[(5-tert-butyl-2-cyclohexylpyrazol-3-yl)methyl]-2-[3-fluoro-4-(methanesulfonamido)phenyl]propanamide |
49804501 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
N-[[5-tert-butyl-2-(3-chlorophenyl)pyrazol-3-yl]methyl]-2-[3-fluoro-4-(methanesulfonamido)phenyl]propanamide |
49804502 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
N-[[5-tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]methyl]-2-[3-fluoro-4-(methanesulfonamido)phenyl]propanamide |
49804506 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
N-[[5-tert-butyl-2-(4-tert-butylphenyl)pyrazol-3-yl]methyl]-2-[3-fluoro-4-(methanesulfonamido)phenyl]propanamide |
49804795 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
N-[[5-tert-butyl-2-(4-chlorophenyl)pyrazol-3-yl]methyl]-2-[3-fluoro-4-(methanesulfonamido)phenyl]propanamide |
49804796 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
(2S)-N-[[5-tert-butyl-2-(4-chlorophenyl)pyrazol-3-yl]methyl]-2-[3-fluoro-4-(methanesulfonamido)phenyl]propanamide |
49804797 |
ChemBL |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
N-[[5-tert-butyl-2-(3-chloro-4-fluorophenyl)pyrazol-3-yl]methyl]-2-[3-fluoro-4-(methanesulfonamido)phenyl]propanamide |
49804798 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
N-(5-(trifluoromethyl)pyrazin-2-yl)-7-(3-(trifluoromethyl)pyridin-2-yl)-1,8-naphthyridin-4-amine |
49863783 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
7-(3-(trifluoromethyl)pyridin-2-yl)-N-(5-(trifluoromethyl)pyrimidin-2-yl)-1,8-naphthyridin-4-amine |
49863784 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
N-(4-chloro-5-(trifluoromethyl)pyrimidin-2-yl)-7-(3-(trifluoromethyl)pyridin-2-yl)-1,8-naphthyridin-4-amine |
49863799 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
5-(Trifluoromethyl)-2-(7-(3-(trifluoromethyl)pyridin-2-yl)-1,8-naphthyridin-4-ylamino)pyrimidine-4-carbonitrile |
49863800 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
5-(Trifluoromethyl)-2-(7-(3-(trifluoromethyl)pyridin-2-yl)-1,8-naphthyridin-4-ylamino)pyrimidine-4-carboxamide |
49863801 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
5-(Trifluoromethyl)-2-(7-(3-(trifluoromethyl)pyridin-2-yl)-1,8-naphthyridin-4-ylamino)pyrimidine-4-carboxylic acid |
49863802 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
4-(trifluoromethyl)-N-(7-(3-(trifluoromethyl)pyridin-2-yl)-1,8-naphthyridin-4-yl)thiazol-2-amine |
49863825 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
N-(5-(trifluoromethyl)pyridin-2-yl)-7-(3-(trifluoromethyl)pyridin-4-yl)-1,8-naphthyridin-4-amine |
49863826 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
N-(5-(trifluoromethyl)pyridin-2-yl)-7-(5-(trifluoromethyl)pyrimidin-4-yl)-1,8-naphthyridin-4-amine |
49863827 |
ChemBL, TTD |