| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-(7-tert-butyl-1-methyl-1,2,3,4-tetrahydroquinolin-4-yl)-3-(1H-indazol-4-yl)urea |
53320280 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
tert-butyl 2-((4-(4-(trifluoromethyl)phenylamino)-7-(3-(trifluoromethyl)pyridin-2-yl)-6,7,8,9-tetrahydro-5H-pyrimido[5,4-d]azepin-2-ylamino)methyl)piperidine-1-carboxylate |
53320485 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
(1R,3S)-4-chloro-5-(4-fluorophenyl)-N-(3-hydroxycyclohexyl)isoxazole-3-carboxamide |
53320830 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
N-cyclopentyl-5-(4-(trifluoromethyl)phenyl)isoxazole-3-carboxamide |
53320831 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-(8-tert-butyl-1-methyl-1,2,3,4-tetrahydroquinolin-4-yl)-3-(1H-indazol-4-yl)urea |
53321243 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
2-(4-(4-(4-(trifluoromethyl)phenylamino)-7-(3-(trifluoromethyl)pyridin-2-yl)-6,7,8,9-tetrahydro-5H-pyrimido[5,4-d]azepin-2-yl)piperazin-1-yl)ethanol |
53321779 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
N2-(2-(dimethylamino)ethyl)-N2-methyl-N4-(4-(trifluoromethyl)phenyl)-7-(3-(trifluoromethyl)pyridin-2-yl)-6,7,8,9-tetrahydro-5H-pyrimido[5,4-d]azepine-2,4-diamine |
53321780 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
2-(3-aminopyrrolidin-1-yl)-N-(4-(trifluoromethyl)phenyl)-7-(3-(trifluoromethyl)pyridin-2-yl)-6,7,8,9-tetrahydro-5H-pyrimido[5,4-d]azepin-4-amine |
53321781 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
N-methyl-N-(1-(4-(4-(trifluoromethyl)phenylamino)-7-(3-(trifluoromethyl)pyridin-2-yl)-6,7,8,9-tetrahydro-5H-pyrimido[5,4-d]azepin-2-yl)pyrrolidin-3-yl)acetamide |
53321782 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
tert-butyl 3-(methyl(4-(4-(trifluoromethyl)phenylamino)-7-(3-(trifluoromethyl)pyridin-2-yl)-6,7,8,9-tetrahydro-5H-pyrimido[5,4-d]azepin-2-yl)amino)piperidine-1-carboxylate |
53321783 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
2-(4-cyclopropylpiperazin-1-yl)-N-(4-(trifluoromethyl)phenyl)-7-(3-(trifluoromethyl)pyridin-2-yl)-6,7,8,9-tetrahydro-5H-pyrimido[5,4-d]azepin-4-amine |
53321847 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
(3H)A778317 |
53321936 |
GtoPDB |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
4-bromo-N-cyclopentyl-5-(4-(trifluoromethoxy)phenyl)isoxazole-3-carboxamide |
53322166 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-(6-tert-butyl-1-methyl-1,2,3,4-tetrahydroquinolin-4-yl)-3-(1H-indazol-4-yl)urea |
53322568 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
(4-Chloro-5-(4-(trifluoromethyl)phenyl)isoxazol-3-yl)(4-hydroxypiperidin-1-yl)methanone |
53322847 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
(1R,3S)-4-chloro-5-(4-fluorophenyl)-N-(3-hydroxycyclopentyl)isoxazole-3-carboxamide |
53322848 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
2-(4-(2-(dimethylamino)ethyl)piperazin-1-yl)-N-(4-(trifluoromethyl)phenyl)-7-(3-(trifluoromethyl)pyridin-2-yl)-6,7,8,9-tetrahydro-5H-pyrimido[5,4-d]azepin-4-amine |
53323109 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
2-(4-isopropylpiperazin-1-yl)-N-(4-(trifluoromethyl)phenyl)-7-(3-(trifluoromethyl)pyridin-2-yl)-6,7,8,9-tetrahydro-5H-pyrimido[5,4-d]azepin-4-amine |
53323161 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
(S)-1-(7-tert-butylchroman-4-yl)-3-(1H-indazol-4-yl)urea |
53323958 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
Cis-(+/-)-4-chloro-N-(3-hydroxycyclohexyl)-5-(4-(trifluoromethyl)phenyl)isoxazole-3-carboxamide |
53324108 |
ChemBL, TTD |