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Drugs And Genes
DRUGs and GENEs
GENE_SYMBOL HGNC_ID UNIPROT_ID DRUG_NAME PUBCHEM_CID Datasource
TRPV1 HGNC:12716 Q8NER1 4-[3-chloro-5-(2-hydroxypropan-2-yl)pyridin-2-yl]-N-[3-fluoro-4-(trifluoromethyl)phenyl]-3,6-dihydro-2H-pyridine-1-carboxamide 57770551 ChemBL
TRPV1 HGNC:12716 Q8NER1 4-[3-chloro-5-[(1R)-1,2-dihydroxyethyl]pyridin-2-yl]-4-fluoro-N-[3-methoxy-4-(trifluoromethyl)phenyl]piperidine-1-carboxamide 57770552 ChemBL
TRPV1 HGNC:12716 Q8NER1 4-[5-[(1R)-1,2-dihydroxyethyl]-3-fluoropyridin-2-yl]-4-fluoro-N-[5-(trifluoromethyl)pyridin-2-yl]piperidine-1-carboxamide 57770553 ChemBL
TRPV1 HGNC:12716 Q8NER1 4-[3-chloro-5-[(1R)-1,2-dihydroxyethyl]pyridin-2-yl]-N-[3-methoxy-4-(trifluoromethyl)phenyl]-3,6-dihydro-2H-pyridine-1-carboxamide 57770554 ChemBL
TRPV1 HGNC:12716 Q8NER1 4-[3-chloro-5-(hydroxymethyl)pyridin-2-yl]-N-[3-phenyl-4-(trifluoromethoxy)phenyl]-3,6-dihydro-2H-pyridine-1-carboxamide 57770566 ChemBL
TRPV1 HGNC:12716 Q8NER1 N-[3-chloro-4-(trifluoromethyl)phenyl]-4-[5-[(1R)-1,2-dihydroxyethyl]-3-fluoropyridin-2-yl]-4-fluoropiperidine-1-carboxamide 57770568 ChemBL
TRPV1 HGNC:12716 Q8NER1 N-[6-(dimethylamino)pyridin-3-yl]-4-phenyl-3-(piperidin-1-ylmethyl)benzamide 57927125 ChemBL, TTD
TRPV1 HGNC:12716 Q8NER1 2-[2-[(E)-2-[4-(trifluoromethoxy)phenyl]ethenyl]-3H-benzimidazol-5-yl]benzenesulfonamide 58381102 ChemBL, TTD
TRPV1 HGNC:12716 Q8NER1 2-[2-[2-[(E)-2-[4-(trifluoromethylsulfonyl)phenyl]ethenyl]-3H-benzimidazol-5-yl]phenyl]propan-2-ol 58381208 ChemBL, TTD
TRPV1 HGNC:12716 Q8NER1 4-borono-N-(4-tert-butyl-phenyl)-benzamide 58639564 ChemBL, TTD
TRPV1 HGNC:12716 Q8NER1 (2R)-N-[(4-tert-butylphenyl)methyl]-2-[3-fluoro-4-(methanesulfonamido)phenyl]propanamide 58755739 ChemBL, TTD
TRPV1 HGNC:12716 Q8NER1 2-[3-fluoro-4-(methanesulfonamido)phenyl]-N-[[2-[4-(4-methoxyphenyl)piperazin-1-yl]-6-(trifluoromethyl)pyridin-3-yl]methyl]propanamide 58873250 ChemBL, TTD
TRPV1 HGNC:12716 Q8NER1 N-[[2-(cyclohexylmethoxy)-6-(trifluoromethyl)pyridin-3-yl]methyl]-2-[3-fluoro-4-(methanesulfonamido)phenyl]propanamide 58873252 ChemBL, TTD
TRPV1 HGNC:12716 Q8NER1 2-[3-fluoro-4-(propan-2-ylsulfonylamino)phenyl]-N-[[2-(4-methylpiperidin-1-yl)-6-(trifluoromethyl)pyridin-3-yl]methyl]propanamide 58873256 ChemBL, TTD
TRPV1 HGNC:12716 Q8NER1 2-[3-fluoro-4-(methanesulfonamido)phenyl]-N-[[2-(pyridin-3-ylmethoxy)-6-(trifluoromethyl)pyridin-3-yl]methyl]propanamide 58873257 ChemBL, TTD
TRPV1 HGNC:12716 Q8NER1 [1-[3-[[2-[3-Fluoro-4-(methanesulfonamido)phenyl]propanoylamino]methyl]-6-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl] acetate 58873260 ChemBL, TTD
TRPV1 HGNC:12716 Q8NER1 [1-[3-[[2-[3-Fluoro-4-(methanesulfonamido)phenyl]propanoylamino]methyl]-6-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl] 2,2-dimethylpropanoate 58873263 ChemBL, TTD
TRPV1 HGNC:12716 Q8NER1 2-[3-fluoro-4-(methanesulfonamido)phenyl]-N-[[2-[(Z)-pent-1-enyl]-6-(trifluoromethyl)pyridin-3-yl]methyl]propanamide 58873266 ChemBL, TTD
TRPV1 HGNC:12716 Q8NER1 2-[3-fluoro-4-(methanesulfonamido)phenyl]-N-[[2-[4-(4-methylphenyl)piperazin-1-yl]-4-(trifluoromethyl)phenyl]methyl]propanamide 58873268 ChemBL, TTD
TRPV1 HGNC:12716 Q8NER1 N-[[6-[chloro(difluoro)methyl]-2-(4-methylpiperidin-1-yl)pyridin-3-yl]methyl]-2-[3-fluoro-4-(methanesulfonamido)phenyl]propanamide 58873274 ChemBL, TTD