| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TRPV3 |
HGNC:18084 |
Q8NET8 |
(2R)-2-[[3-fluoro-6-(2,4,5-trifluorophenyl)pyridin-2-yl]methylamino]-3-methylbutan-1-ol |
68312879 |
ChemBL |
| TRPV3 |
HGNC:18084 |
Q8NET8 |
(2R)-2-[[3-fluoro-6-(5-fluoro-3,4-dihydro-1H-isoquinolin-2-yl)pyridin-2-yl]methylamino]-3-methylbutan-1-ol |
68312890 |
ChemBL |
| TRPV3 |
HGNC:18084 |
Q8NET8 |
3-[[2-[4-(Trifluoromethyl)phenyl]pyrimidin-4-yl]methylamino]butan-2-ol |
68312895 |
ChemBL |
| TRPV3 |
HGNC:18084 |
Q8NET8 |
(3R)-3-[[3-fluoro-6-[6-(trifluoromethyl)pyridin-3-yl]pyridin-2-yl]methylamino]-2,4-dimethylpentan-2-ol |
68312898 |
ChemBL |
| TRPV3 |
HGNC:18084 |
Q8NET8 |
(2R)-2-[[6-(2-cyclohexylethynyl)-3-fluoropyridin-2-yl]methylamino]-3-methylbutan-1-ol |
68312902 |
ChemBL |
| TRPV3 |
HGNC:18084 |
Q8NET8 |
(3R)-3-({[5-fluoro-6'-(trifluoromethyl)-2,3'-bipyridin-6-yl]methyl}amino)-4-methylpentan-2-ol |
68312912 |
ChemBL |
| TRPV3 |
HGNC:18084 |
Q8NET8 |
(2R)-2-[[3-fluoro-6-[1-(4-fluorophenyl)ethyl]pyridin-2-yl]methylamino]-3-methylbutan-1-ol |
68312930 |
ChemBL |
| TRPV3 |
HGNC:18084 |
Q8NET8 |
(2R)-2-[[3-chloro-6-[6-(trifluoromethyl)pyridin-3-yl]pyridin-2-yl]methylamino]-3-methylbutan-1-ol |
68312944 |
ChemBL |
| TRPV3 |
HGNC:18084 |
Q8NET8 |
(2R)-3,3-dimethyl-2-[[2-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]methylamino]butan-1-ol |
68312949 |
ChemBL |
| TRPV3 |
HGNC:18084 |
Q8NET8 |
(2R)-2-[[3-fluoro-6-[4-(trifluoromethyl)phenyl]pyridin-2-yl]methylamino]-3-methylbutan-1-ol |
68312982 |
ChemBL |
| TRPV3 |
HGNC:18084 |
Q8NET8 |
(2R)-2-[[3-fluoro-6-[4-(trifluoromethoxy)phenyl]pyridin-2-yl]methylamino]-3-methylbutan-1-ol |
68312988 |
ChemBL |
| TRPV3 |
HGNC:18084 |
Q8NET8 |
(2R)-2-[[2-(4-chlorophenyl)pyrimidin-4-yl]methylamino]-3-methylbutan-1-ol |
68312996 |
ChemBL |
| TRPV3 |
HGNC:18084 |
Q8NET8 |
N-benzyl-3-[5-fluoro-6-[[[(2R)-1-hydroxy-3-methylbutan-2-yl]amino]methyl]pyridin-2-yl]-N-methylbenzamide |
68312997 |
ChemBL |
| TRPV3 |
HGNC:18084 |
Q8NET8 |
(2R)-2-[[3-fluoro-6-[2-(2,2,2-trifluoroethoxy)pyrimidin-5-yl]pyridin-2-yl]methylamino]-3-methylbutan-1-ol |
68313003 |
ChemBL |
| TRPV3 |
HGNC:18084 |
Q8NET8 |
(2R)-2-({[3-fluoro-6-(2,3,4-trifluorophenyl)pyridin-2-yl]methyl}amino)-3-methylbutan-1-ol |
68313015 |
ChemBL |
| TRPV3 |
HGNC:18084 |
Q8NET8 |
(2R)-2-[[3-fluoro-6-(3-pyrrolidin-1-ylsulfonylphenyl)pyridin-2-yl]methylamino]-3-methylbutan-1-ol |
68313017 |
ChemBL |
| TRPV3 |
HGNC:18084 |
Q8NET8 |
(2R)-2-[[3-fluoro-6-(5-methylthiophen-2-yl)pyridin-2-yl]methylamino]-3-methylbutan-1-ol |
68313046 |
ChemBL |
| TRPV3 |
HGNC:18084 |
Q8NET8 |
TRPV3 antagonist 74a |
71554840 |
ChemBL, TTD |
| TRPV3 |
HGNC:18084 |
Q8NET8 |
[3-[[6-[4-(Trifluoromethyl)phenyl]pyridin-2-yl]methylamino]-2-bicyclo[2.2.1]heptanyl]methanol |
77475706 |
ChemBL |
| TRPV3 |
HGNC:18084 |
Q8NET8 |
N1-[4-(2,3-Difluoro-4-trifluoromethylphenyl)-1,3-thiazol-2-yl]-2-(1,3,6-trimethyl-2,4-dioxo-1,2,3,4-tetrahydrofuro[2,3-d]pyrimidin-5-yl)acetamide |
86666696 |
ChemBL |