| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[6-[2-(4-fluorophenyl)ethynyl]-8-(2-methylpropylamino)imidazo[1,2-a]pyrazin-3-yl]benzamide |
54767993 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
US9555022, Example 02.09 |
54768802 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
US9555022, Example 02.17 |
54769502 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
US9555022, Example 02.29 |
54770142 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
US9555022, Example 02.44 |
54770807 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
8-[2-methoxy-4-[(1-methylpiperidin-4-yl)carbamoyl]anilino]-4,4-dimethyl-5H-[1,2]oxazolo[4,3-h]quinazoline-3-carboxamide |
56645226 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
8-[2-methoxy-4-[(1-methylpiperidin-4-yl)carbamoyl]anilino]-5,5-dimethyl-4H-[1,2]oxazolo[4,5-h]quinazoline-3-carboxamide |
56645845 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[(1R)-2-amino-1-phenylethyl]-8-[2-methoxy-4-[(1-methylpiperidin-4-yl)carbamoyl]anilino]-5,5-dimethyl-4H-[1,2]oxazolo[4,5-h]quinazoline-3-carboxamide |
56646033 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
5-Chloro-4-(1H-indol-3-yl)-N-(2-methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)phenyl)pyrimidin-2-amine |
56655374 |
DSigDB |
| TTK |
HGNC:12401 |
P33981 |
N-(2,6-diethylphenyl)-1-methyl-8-[4-[(2R)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]-2-(trifluoromethoxy)anilino]-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide |
56659726 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
N-(2,6-diethylphenyl)-8-[4-[4-(dimethylamino)piperidine-1-carbonyl]-2-(trifluoromethoxy)anilino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide |
56663194 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
8-anilino-N-(2,6-diethylphenyl)-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide |
56666592 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
8-[4-carbamoyl-2-(trifluoromethoxy)anilino]-N-(2,6-diethylphenyl)-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide |
56676834 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
N-(2,6-diethylphenyl)-8-[4-[2-(dimethylamino)ethylcarbamoyl]-2-(trifluoromethoxy)anilino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide |
56676835 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
N-(2,6-diethylphenyl)-1-methyl-8-[4-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]-2-(trifluoromethoxy)anilino]-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide |
56676891 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
4-(2-Amino-5-{4-[(Dimethylamino)methyl]thiophen-2-Yl}pyridin-3-Yl)-2-{(1r)-1-[2-(Trifluoromethyl)phenyl]ethoxy}benzamide |
56947168 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
4-(2-Amino-5-{4-[(dimethylamino)methyl]thiophen-2-YL}pyridin-3-YL)-2-{[(1R,2Z)-4,4,4-trifluoro-1-methylbut-2-EN-1-YL]oxy}benzamide |
56947170 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
9-Cyclopentyl-2-[[2-methoxy-4-[(1-methylpiperidin-4-yl)oxy]-phenyl]amino]-7-methyl-7,9-dihydro-8H-purin-8-one |
56973724 |
ChemBL, GtoPDB, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-(8-((2-hydroxyethyl)amino)imidazo[1,2-a]pyrazin-3-yl)benzamide |
57379118 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-Cyclopropyl-4-[8-[(phenylmethyl)amino]imidazo[1,2-a]pyrazin-3-yl]benzamide |
57379119 |
ChemBL, TTD |