| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TTK |
HGNC:12401 |
P33981 |
TC-Mps1-12 |
70682875 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-(2-methyl-4-morpholin-4-ylphenyl)-6-morpholin-4-yl-7H-purin-2-amine |
70684107 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
[4-[4-[[6-(cyclohexylamino)-7H-purin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-(4-hydroxycyclohexyl)methanone |
70684108 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
6-(cyclohexylmethyl)-N-(2-methyl-4-morpholin-4-ylphenyl)-7H-purin-2-amine |
70686248 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
6-N-cyclohexyl-2-N-[4-[4-(diethylaminomethyl)piperidin-1-yl]-2-methoxyphenyl]-7H-purine-2,6-diamine |
70686252 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
2-[1-[4-[[6-(cyclohexylamino)-7H-purin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]-1-(4-methylpiperazin-1-yl)ethanone |
70688373 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
2-[1-[4-[[6-(cyclohexylamino)-7H-purin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]-1-[3-(dimethylamino)pyrrolidin-1-yl]ethanone |
70688374 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
[1-[4-[[6-(cyclohexylamino)-7H-purin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]-(3-hydroxyazetidin-1-yl)methanone |
70688375 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
2-N-(2-methyl-4-morpholin-4-ylphenyl)-6-N-piperidin-4-yl-7H-purine-2,6-diamine |
70690388 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
[4-[4-[[6-(cyclohexylamino)-7H-purin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-(4-methylpiperazin-1-yl)methanone |
70692558 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
6-N-cyclohexyl-2-N-(2-methylsulfanyl-4-morpholin-4-ylphenyl)-7H-purine-2,6-diamine |
70694608 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
2-[4-[4-[[6-(cyclohexylamino)-7H-purin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-N-methyl-2-oxoacetamide |
70696648 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
[1-[4-[[6-(cyclohexylamino)-7H-purin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]-[3-(dimethylamino)pyrrolidin-1-yl]methanone |
70696649 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
18-Fluoro-25-methoxy-31-methyl-22,22-dioxo-3,22lambda6,30-trithia-6,8,15,23,26-pentazahexacyclo[22.3.1.12,5.110,13.117,21.04,9]hentriaconta-1(28),2(31),4,6,8,10,12,17,19,21(29),24,26-dodecaen-16-one |
71041971 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[3-(4-morpholin-4-ylphenyl)-1H-indazol-5-yl]-2-pyrrolidin-1-yl-2-thiophen-3-ylacetamide |
71549884 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
3-[4-(4-hydroxypiperidin-1-yl)phenyl]-N-[(1-morpholin-4-ylcyclohexyl)methyl]-1H-indazole-5-carboxamide |
71550158 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
5-[5-Ethoxy-6-(1-Methyl-1h-Pyrazol-4-Yl)-1h-Indazol-3-Yl]-2-Methylbenzenesulfonamide |
71576779 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
US9663510, Example 01.07 |
71577161 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
Empesertib |
71599640 |
ChemBL, GtoPDB, Pubchem, TTD |
| TTK |
HGNC:12401 |
P33981 |
US9663510, Example 01.09 |
71599805 |
ChemBL |