| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TTK |
HGNC:12401 |
P33981 |
N-[4-(2,3-dimethylimidazol-4-yl)-2-methoxyphenyl]-6-[1-(oxan-4-yl)pyrazol-4-yl]isoquinolin-3-amine |
73388611 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[4-(2,3-dimethylimidazol-4-yl)-2-methoxyphenyl]-6-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]isoquinolin-3-amine |
73388688 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
1-[4-[7-[2-Ethoxy-4-(4-methyl-1,2,4-triazol-3-yl)anilino]-1,6-naphthyridin-2-yl]pyrazol-1-yl]-2-methylpropan-2-ol |
73388689 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
1-[4-[7-[2-Methoxy-4-(4-methyl-1,2,4-triazol-3-yl)anilino]-1,6-naphthyridin-2-yl]pyrazol-1-yl]-2-methylpropan-2-ol |
73388690 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
[3-(Difluoromethoxy)-4-[[6-[1-(2-hydroxy-2-methylpropyl)pyrazol-4-yl]isoquinolin-3-yl]amino]phenyl]-(3-methoxyazetidin-1-yl)methanone |
73388691 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
1-[[4-[7-[4-(2,3-Dimethylimidazol-4-yl)-2-methoxyanilino]-1,6-naphthyridin-2-yl]pyrazol-1-yl]methyl]cyclobutan-1-ol |
73388692 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
1-[4-[3-[2-Ethoxy-4-(4-methyl-1,2,4-triazol-3-yl)anilino]isoquinolin-6-yl]pyrazol-1-yl]-2-methylpropan-2-ol |
73388693 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
1-[4-[3-[4-(2,3-Dimethylimidazol-4-yl)-3-fluoro-2-methoxyanilino]isoquinolin-6-yl]pyrazol-1-yl]-2-methylpropan-2-ol |
73388694 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
1-[4-[3-[2-Methoxy-4-(1-methylpyrazol-4-yl)anilino]isoquinolin-6-yl]pyrazol-1-yl]-2-methylpropan-2-ol |
73388695 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
1-[4-[3-(4-Fluoro-2-methoxyanilino)isoquinolin-6-yl]pyrazol-1-yl]-2-methylpropan-2-ol |
73388696 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
(2R)-1-[4-[3-[4-(2,3-dimethylimidazol-4-yl)-2-methoxyanilino]isoquinolin-6-yl]pyrazol-1-yl]propan-2-ol |
73388697 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
(3,3-Difluoroazetidin-1-yl)-[4-[[6-[1-(2-hydroxy-2-methylpropyl)pyrazol-4-yl]isoquinolin-3-yl]amino]-3-methoxyphenyl]methanone |
73388769 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
[3-Ethoxy-4-[[6-[1-(2-hydroxy-2-methylpropyl)pyrazol-4-yl]isoquinolin-3-yl]amino]phenyl]-(3-methoxyazetidin-1-yl)methanone |
73388770 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
[4-[[6-[1-(2-Hydroxy-2-methylpropyl)pyrazol-4-yl]isoquinolin-3-yl]amino]-3-methoxyphenyl]-(6-oxa-2-azaspiro[3.4]octan-2-yl)methanone |
73388771 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
1-[4-[[6-[1-(2-Hydroxy-2-methylpropyl)pyrazol-4-yl]isoquinolin-3-yl]amino]-3-methoxybenzoyl]piperidine-4-carbonitrile |
73388772 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
1-[4-[3-[2-Chloro-4-(5-methyl-1,3,4-oxadiazol-2-yl)anilino]isoquinolin-6-yl]pyrazol-1-yl]-2-methylpropan-2-ol |
73388773 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
(2S)-1-[4-[3-[4-(2,3-dimethylimidazol-4-yl)-2-methoxyanilino]isoquinolin-6-yl]pyrazol-1-yl]propan-2-ol |
73388774 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
[4-[[6-[1-(2,3-Dimethoxypropyl)pyrazol-4-yl]isoquinolin-3-yl]amino]-3-methoxyphenyl]-(3-methoxyazetidin-1-yl)methanone |
73388852 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
5-[4-[[6-[1-(2-Hydroxy-2-methylpropyl)pyrazol-4-yl]isoquinolin-3-yl]amino]-3-methoxyphenyl]-1-methylimidazole-2-carbonitrile |
73388853 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
US10188642, Example 83 |
73388854 |
ChemBL |