| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[5-(2,3-difluoro-4-methoxyphenoxy)-7-(3,3,3-trifluoropropylamino)pyrazolo[1,5-a]pyrimidin-3-yl]-2-methylbenzamide |
156015586 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
1-Methyl-3-[4-[8-(2-methylpropylamino)imidazo[1,2-a]pyrazin-3-yl]phenyl]urea |
156015816 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-(4-fluorophenyl)-N-[4-[2-(2-methoxy-4-methylsulfonylanilino)-[1,2,4]triazolo[1,5-a]pyridin-6-yl]phenyl]butanamide |
156016456 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[6-(4-hydroxy-3,5-dimethylphenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]-6-oxopyran-3-carboxamide |
156016785 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-2-methyl-4-[6-(2-phenylethyl)-8-(3,3,3-trifluoropropylamino)imidazo[1,2-a]pyrazin-3-yl]benzamide |
156018550 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[8-[(3-hydroxy-3-methylcyclobutyl)methylamino]-6-pyridin-3-yloxyimidazo[1,2-b]pyridazin-3-yl]-2-methylbenzamide |
156018633 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
6-[8-(2-Methylpropylamino)imidazo[1,2-a]pyrazin-3-yl]isoquinolin-1-amine |
156019062 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[6-(4-hydroxy-3,5-dimethylphenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]thiophene-2-carboxamide |
156019741 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-benzyl-4-[2-(2-cyanoanilino)-[1,2,4]triazolo[1,5-a]pyridin-6-yl]benzamide |
156021553 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2,6-Dimethyl-4-[2-(1-phenylethylamino)-[1,2,4]triazolo[1,5-a]pyridin-6-yl]phenol |
156021588 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[4-(2-methylpropylamino)imidazo[2,1-f][1,2,4]triazin-7-yl]benzamide |
156021987 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
3-(3-amino-1H-indazol-6-yl)-N-(2-methylpropyl)imidazo[1,2-a]pyrazin-8-amine |
156022070 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-(2,6-diethylphenyl)-2-[4-(4-methylpiperazin-1-yl)-2-(propanoylamino)anilino]-5,6-dihydropyrimido[4,5-e]indolizine-7-carboxamide |
162639277 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
TTK inhibitor 3 |
162640906 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-(2,6-diethylphenyl)-2-[4-(4-methylpiperazin-1-yl)-2-(prop-2-enoylamino)anilino]-5,6-dihydropyrimido[4,5-e]indolizine-7-carboxamide |
163196379 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[4-[2-[2-methoxy-4-(4-methylpiperazin-1-yl)anilino]-5-methyl-7-oxopyrido[2,3-d]pyrimidin-8-yl]cyclohexyl]cyclopentanecarboxamide |
164609243 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[4-[2-[2-methoxy-4-(4-methylpiperazin-1-yl)anilino]-5-methyl-7-oxopyrido[2,3-d]pyrimidin-8-yl]cyclohexyl]-2,2-dimethylpropanamide |
164609376 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-[2-Methoxy-4-(4-methylpiperazin-1-yl)anilino]-5-methyl-8-(1-propanoylazetidin-3-yl)pyrido[2,3-d]pyrimidin-7-one |
164610281 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-[2-methoxy-4-(4-methylpiperazin-1-yl)anilino]-5-methyl-8-[(3S)-1-propanoylpyrrolidin-3-yl]pyrido[2,3-d]pyrimidin-7-one |
164614031 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-[2-methoxy-4-(4-methylpiperazin-1-yl)anilino]-5-methyl-8-[(3R)-1-propanoylpiperidin-3-yl]pyrido[2,3-d]pyrimidin-7-one |
164614085 |
ChemBL |