| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TYK2 |
HGNC:12440 |
P29597 |
Brepocitinib |
118878093 |
DGidb, GtoPDB, Pubchem |
| TYK2 |
HGNC:12440 |
P29597 |
US9663526, Example 94 |
118878190 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
US10463675, Example 95 |
118878248 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
Jak1/tyk2-IN-1 |
118878262 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
(3-amino-1H-indazol-5-yl)-[(2S)-2-(4-chlorophenyl)pyrrolidin-1-yl]methanone |
118879520 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
US10081635, Example 5 |
118911481 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
US10081635, Example 41 |
118911570 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-(2-carbamoylanilino)-N-ethyl-6-[(5-fluoropyridin-2-yl)amino]pyridine-3-carboxamide |
121284861 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-(4-carbamoyl-2-methoxyanilino)-6-[(5-fluoropyridin-2-yl)amino]-N-methylpyridine-3-carboxamide |
121284991 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
6-[(5-fluoropyridin-2-yl)amino]-4-(2-methoxyanilino)-N-methylpyridine-3-carboxamide |
121285043 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
6-({4-[(3S)-3-cyano-3-cyclopropyl-2-oxopyrrolidin-1-yl]pyridin-2-yl}amino)-N,N-dimethylpyridine-3-carboxamide |
121374385 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
Xmu-MP-1 |
121499143 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
4-[(1-benzylpiperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-5-carboxamide |
122182157 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
6-bromo-2-(1-methyl-3-propan-2-ylpyrazol-4-yl)-7-[4-(pyridin-3-ylmethyl)piperazin-1-yl]-1H-imidazo[4,5-b]pyridine |
122189151 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N,N-dicyclopropyl-10-ethyl-3-methyl-7-(methylamino)-3,5,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-1,4,6,8,11-pentaene-11-carboxamide |
122191618 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
2-methoxyethyl N-[11-(dicyclopropylcarbamoyl)-10-ethyl-3-methyl-3,5,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-1,4,6,8,11-pentaen-7-yl]carbamate |
122191619 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N,N-dicyclopropyl-10-ethyl-7-(2-methoxyethylcarbamoylamino)-3-methyl-3,5,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-1,4,6,8,11-pentaene-11-carboxamide |
122191620 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N,N-dicyclopropyl-7-[(2,5-dimethylpyrazol-3-yl)amino]-10-ethyl-3-methyl-3,5,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-1,4,6,8,11-pentaene-11-carboxamide |
122191625 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-[1-(oxiran-2-ylmethyl)triazol-4-yl]-7H-pyrrolo[2,3-d]pyrimidine |
122191778 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
2-(2-Aminoethyl)-1-(3-aminopropyl)benzimidazole-5-carboxamide |
122192065 |
ChemBL, TTD |