| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TYK2 |
HGNC:12440 |
P29597 |
(~{E})-3-[5-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)furan-2-yl]prop-2-enenitrile |
134611727 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
3-[5-(3-Cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)furan-2-yl]propanenitrile |
134611728 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
6-[(3,5-difluoro-2-methoxyphenyl)amino]-N-(3,4-dihydroxy-3-methylbutyl)-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide |
134611892 |
DGidb, GtoPDB |
| TYK2 |
HGNC:12440 |
P29597 |
4-({4-[(1S,4S)-5-(cyanoacetyl)-2,5-diazabicyclo[2.2.1]heptan-2-yl]pyrimidin-2-yl}amino)-N-ethylbenzamide |
134812674 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
Deucravacitinib |
134821691 |
ChemBL, DGidb, GtoPDB, Pubchem, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
((S)-2,2-difluorocyclopropyl)(3-(2-((1-methyl-1H-pyrazol-4-yl)amino)pyrimidin-4-yl)-3,8-diazabicyclo[3.2.1]octan-8-yl)methanone |
135087198 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
3-(4-cyano-3-methoxyanilino)-1-[(3R,4S)-4-cyanooxan-3-yl]pyrazole-4-carboxamide |
135125189 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
Atinvicitinib |
135138184 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
1-Cyclopropyl-3-(3-(5-(morpholinomethyl)-1H-benzo[d]imidazol-2-yl)-1H-pyrazol-4-yl)urea |
135398495 |
ChemBL, DGidb, Pubchem, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
Otssp167 |
135398499 |
DSigDB |
| TYK2 |
HGNC:12440 |
P29597 |
Dovitinib |
135398510 |
DGidb, Pubchem |
| TYK2 |
HGNC:12440 |
P29597 |
Indirubin E804 |
135398511 |
DSigDB |
| TYK2 |
HGNC:12440 |
P29597 |
Rg-1530 |
135398512 |
DGidb |
| TYK2 |
HGNC:12440 |
P29597 |
Hesperadin |
135421442 |
ChemBL, DGidb |
| TYK2 |
HGNC:12440 |
P29597 |
Nintedanib |
135423438 |
Pubchem |
| TYK2 |
HGNC:12440 |
P29597 |
4-[(4-Aminocyclohexyl)amino]-3-(1h-Benzimidazol-2-Yl)-1h-Pyridin-2-One |
135567142 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-[3-(1h-Benzimidazol-2-Yl)-1h-Indazol-6-Yl]-3-Ethylphenol |
135567293 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
6-(2-Ethyl-4-Hydroxyphenyl)-1h-Indazole-3-Carboxamide |
135567294 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
6-(2-Ethyl-4-Hydroxyphenyl)-N-(6-Methylpyridin-3-Yl)-1h-Indazole-3-Carboxamide |
135567295 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
PF-06263276 |
135567296 |
ChemBL, DGidb, GtoPDB, TTD |