| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TYK2 |
HGNC:12440 |
P29597 |
2-[4-[[5-Carbamoyl-2-(2,6-difluorophenyl)pyrimidin-4-yl]amino]phenyl]acetic acid |
168268990 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
6-(cyclopropanecarbonylamino)-4-[3-[(2-cyclopropyl-1-oxo-3H-isoindol-5-yl)carbamoyl]-2-methoxyanilino]-N-(trideuteriomethyl)pyridazine-3-carboxamide |
168269195 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
4-[3-[[4-[[(2S)-1,4-dioxan-2-yl]methylamino]phenyl]carbamoyl]-2-methoxyanilino]-6-(pyridin-2-ylamino)-N-(trideuteriomethyl)pyridazine-3-carboxamide |
168271265 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
4-[3-[(5-carbamoylthiophen-3-yl)carbamoyl]-2-methoxyanilino]-6-(cyclopropanecarbonylamino)-N-(trideuteriomethyl)pyridazine-3-carboxamide |
168271274 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
4-[3-[(4-carbamoylphenyl)carbamoyl]-2-methoxyanilino]-6-(cyclopropanecarbonylamino)-N-(trideuteriomethyl)pyridazine-3-carboxamide |
168272862 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
6-(cyclopropanecarbonylamino)-4-[2-methoxy-3-[(2-oxo-1,3-dihydroindol-5-yl)carbamoyl]anilino]-N-(trideuteriomethyl)pyridazine-3-carboxamide |
168274441 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
6-(cyclopropanecarbonylamino)-4-[2-methoxy-3-[[4-(pyrrolidine-1-carbonyl)cyclohexyl]carbamoyl]anilino]-N-(trideuteriomethyl)pyridazine-3-carboxamide |
168274546 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
6-(cyclopropanecarbonylamino)-4-[2-methoxy-3-[[4-(oxan-4-ylmethylamino)phenyl]carbamoyl]anilino]-N-(trideuteriomethyl)pyridazine-3-carboxamide |
168276191 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
6-(cyclopropanecarbonylamino)-4-[3-[[4-(diethylcarbamoyl)phenyl]carbamoyl]-2-methoxyanilino]-N-(trideuteriomethyl)pyridazine-3-carboxamide |
168277472 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
4-[3-[(5-carbamoylpyridin-2-yl)carbamoyl]-2-methoxyanilino]-6-(cyclopropanecarbonylamino)-N-(trideuteriomethyl)pyridazine-3-carboxamide |
168277565 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
6-(cyclopropanecarbonylamino)-4-[3-[[4-(ethylcarbamoyl)phenyl]carbamoyl]-2-methoxyanilino]-N-(trideuteriomethyl)pyridazine-3-carboxamide |
168278744 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
2-(2,6-difluorophenyl)-4-[4-[(3S)-3-hydroxypyrrolidine-1-carbonyl]anilino]-6,7-dihydropyrrolo[3,4-b]pyridin-5-one |
168279494 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
4-[3-[[4-(cyclopentylcarbamoyl)phenyl]carbamoyl]-2-methoxyanilino]-6-(cyclopropanecarbonylamino)-N-(trideuteriomethyl)pyridazine-3-carboxamide |
168280054 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
4-[3-[[4-(7-azabicyclo[2.2.1]heptane-7-carbonyl)phenyl]carbamoyl]-2-methoxyanilino]-6-(cyclopropanecarbonylamino)-N-(trideuteriomethyl)pyridazine-3-carboxamide |
168280582 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
6-(cyclopropanecarbonylamino)-4-[3-[[3-fluoro-4-(pyrrolidine-1-carbonyl)phenyl]carbamoyl]-2-methoxyanilino]-N-(trideuteriomethyl)pyridazine-3-carboxamide |
168281199 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
6-(cyclopropanecarbonylamino)-4-[2-methoxy-3-[(3-oxo-1,2-dihydroisoindol-4-yl)carbamoyl]anilino]-N-(trideuteriomethyl)pyridazine-3-carboxamide |
168281331 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
N-[5-[2-[(1R)-2,2-difluorocyclopropanecarbonyl]-2-azaspiro[4.5]decan-8-yl]-[1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide |
168282756 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
6-(cyclopropanecarbonylamino)-4-[2-methoxy-3-[[4-(methylcarbamoyl)phenyl]carbamoyl]anilino]-N-(trideuteriomethyl)pyridazine-3-carboxamide |
168283269 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
2-(2,6-Difluorophenyl)-4-[[5-(pyrrolidine-1-carbonyl)pyridin-2-yl]amino]-6,7-dihydropyrrolo[3,4-b]pyridin-5-one |
168284796 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
6-(cyclopropanecarbonylamino)-4-[2-methoxy-3-[[4-(pyrrolidine-1-carbonyl)phenyl]carbamoyl]anilino]-N-(trideuteriomethyl)pyridazine-3-carboxamide |
168285545 |
ChemBL |