| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| USP25 |
HGNC:12624 |
Q9UHP3 |
3-amino-N-[2-(2,5-difluoro-4-piperazin-1-ylphenyl)ethyl]-5-fluoro-6-methoxythieno[2,3-b]pyridine-2-carboxamide |
155567524 |
ChemBL |
| USP25 |
HGNC:12624 |
Q9UHP3 |
3-amino-N-[2-(2-fluoro-4-piperazin-1-ylphenyl)ethyl]-6-methylthieno[2,3-b]pyridine-2-carboxamide |
155567843 |
ChemBL |
| USP25 |
HGNC:12624 |
Q9UHP3 |
3-amino-N-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-2-fluorophenyl]ethyl]-6-methylthieno[2,3-b]pyridine-2-carboxamide |
155568058 |
ChemBL |
| USP25 |
HGNC:12624 |
Q9UHP3 |
3-amino-6-methyl-N-[(2S)-2-(4-piperazin-1-ylphenyl)propyl]thieno[2,3-b]pyridine-2-carboxamide;hydrochloride |
155568433 |
ChemBL |
| USP25 |
HGNC:12624 |
Q9UHP3 |
3-amino-6-methyl-N-[2-[4-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)phenyl]ethyl]thieno[2,3-b]pyridine-2-carboxamide |
155568531 |
ChemBL |
| USP28 |
HGNC:12625 |
Q96RU2 |
USP25/28 inhibitor AZ1 |
135397656 |
ChemBL |
| USP28 |
HGNC:12625 |
Q96RU2 |
7-amino-N-[(2S)-2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-3-fluorophenyl]propyl]-3-methylthieno[2,3-b]pyrazine-6-carboxamide |
139578253 |
ChemBL |
| USP28 |
HGNC:12625 |
Q96RU2 |
7-amino-N-[(2R)-2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-3-fluorophenyl]propyl]-3-methylthieno[2,3-b]pyrazine-6-carboxamide |
139578264 |
ChemBL |
| USP28 |
HGNC:12625 |
Q96RU2 |
7-amino-3-methyl-N-[2-(4-piperazin-1-ylphenyl)ethyl]thieno[2,3-b]pyrazine-6-carboxamide |
139578266 |
ChemBL |
| USP28 |
HGNC:12625 |
Q96RU2 |
3-amino-6-[(1R)-1-hydroxyethyl]-N-[2-(4-piperazin-1-ylphenyl)ethyl]thieno[2,3-b]pyridine-2-carboxamide |
141734477 |
ChemBL |
| USP28 |
HGNC:12625 |
Q96RU2 |
3-amino-N-[2-[2,5-difluoro-4-[3-(methylamino)azetidin-1-yl]phenyl]ethyl]-6-methylthieno[2,3-b]pyridine-2-carboxamide |
141734478 |
ChemBL |
| USP28 |
HGNC:12625 |
Q96RU2 |
3-amino-N-[2-[2,5-difluoro-4-[(3S,4S)-3-fluoro-4-(methylamino)pyrrolidin-1-yl]phenyl]ethyl]-6-methylthieno[2,3-b]pyridine-2-carboxamide |
141734483 |
ChemBL |
| USP28 |
HGNC:12625 |
Q96RU2 |
3-amino-N-[2-[2,5-difluoro-4-[(3R)-3-methylpiperazin-1-yl]phenyl]ethyl]-6-methylthieno[2,3-b]pyridine-2-carboxamide |
141734494 |
ChemBL |
| USP28 |
HGNC:12625 |
Q96RU2 |
3-amino-6-methoxy-N-[2-(4-piperazin-1-ylphenyl)ethyl]thieno[2,3-b]pyridine-2-carboxamide |
141734503 |
ChemBL |
| USP28 |
HGNC:12625 |
Q96RU2 |
3-amino-6-methyl-N-[2-[4-[(3S)-3-methylpiperazin-1-yl]phenyl]ethyl]thieno[2,3-b]pyridine-2-carboxamide |
141734514 |
ChemBL |
| USP28 |
HGNC:12625 |
Q96RU2 |
3-amino-N-[2-[2,5-difluoro-4-[(3R,4R)-3-fluoro-4-(methylamino)pyrrolidin-1-yl]phenyl]ethyl]-6-methylthieno[2,3-b]pyridine-2-carboxamide |
141734515 |
ChemBL |
| USP28 |
HGNC:12625 |
Q96RU2 |
3-amino-6-methyl-N-[2-(4-piperazin-1-yl-3-pyridin-2-ylphenyl)ethyl]thieno[2,3-b]pyridine-2-carboxamide |
141734524 |
ChemBL |
| USP28 |
HGNC:12625 |
Q96RU2 |
3-amino-N-[2-(2,5-difluoro-4-piperazin-1-ylphenyl)ethyl]-6-methylthieno[2,3-b]pyridine-2-carboxamide |
141734528 |
ChemBL |
| USP28 |
HGNC:12625 |
Q96RU2 |
3-amino-N-[2-[4-(6,8-dihydro-5H-imidazo[1,2-a]pyrazin-7-yl)phenyl]ethyl]-6-methylthieno[2,3-b]pyridine-2-carboxamide |
141734540 |
ChemBL |
| USP28 |
HGNC:12625 |
Q96RU2 |
3-amino-N-[2-(3-fluoro-4-piperazin-1-ylphenyl)ethyl]-6-methylthieno[2,3-b]pyridine-2-carboxamide;hydrochloride |
141734542 |
ChemBL |