GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
YES1 |
HGNC:12841 |
P07947 |
2-(4-(2-(1H-imidazol-1-yl)ethoxy)phenyl)-4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridine |
10294883 |
DGidb |
YES1 |
HGNC:12841 |
P07947 |
(R)-6-(4-((4-Ethylpiperazin-1-yl)methyl)phenyl)-N-(1-phenylethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine |
10297043 |
ChemBL, Pubchem, TTD |
YES1 |
HGNC:12841 |
P07947 |
N-(5-chloro-2H-1,3-benzodioxol-4-yl)-5-(oxan-4-yloxy)-7-[3-(pyrrolidin-1-yl)propoxy]quinazolin-4-amine |
10301884 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
Saracatinib |
10302451 |
ChemBL, DGidb, DSigDB, GtoPDB, Pubchem, TTD |
YES1 |
HGNC:12841 |
P07947 |
3-[2-[(Z)-[5-(methylsulfamoyl)-2-oxo-1H-indol-3-ylidene]methyl]-4,5,6,7-tetrahydro-1H-indol-3-yl]propanamide |
10320381 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
7-(2,6-dimethylphenyl)-N-phenylbenzo[e][1,2,4]triazin-3-amine |
10404115 |
ChemBL |
YES1 |
HGNC:12841 |
P07947 |
5-Ethanesulfonyl-3-[1-{3-[3-(4-methyl-piperazin-1-yl)-propyl]-4,5,6,7-tetrahydro-1H-indol-2-yl}-meth-(Z)-ylidene]-1,3-dihydro-indol-2-one |
10413508 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
Tesevatinib |
10458325 |
ChemBL, Pubchem |
YES1 |
HGNC:12841 |
P07947 |
[4-(3-{2-[5-Methylsulfamoyl-2-oxo-1,2-dihydro-indol-(3Z)-ylidenemethyl]-4,5,6,7-tetrahydro-1H-indol-3-yl}-propyl)-piperazin-1-yl]-acetic acid |
10482445 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
(S)-5-(3-Fluorophenyl)-N-(piperidin-3-yl)-3-ureidothiophene-2-carboxamide |
11152667 |
ChemBL, DGidb, DSigDB, Pubchem |
YES1 |
HGNC:12841 |
P07947 |
N-(2-Chloro-6-methylphenyl)-2-((2,6-dimethyl-4-pyrimidinyl)amino)-5-thiazolecarboxamide |
11153014 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
5-methyl-7-(3-phenoxyphenyl)-N-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amine |
11155941 |
DGidb |
YES1 |
HGNC:12841 |
P07947 |
Sdccggsk-0000152.P001 |
11163861 |
DGidb |
YES1 |
HGNC:12841 |
P07947 |
Regorafenib |
11167602 |
DGidb, DSigDB |
YES1 |
HGNC:12841 |
P07947 |
Tamatinib |
11213558 |
DGidb, DSigDB |
YES1 |
HGNC:12841 |
P07947 |
N-benzyl-1-(2-chloro-2-phenyl-ethyl)pyrazolo[3,4-d]pyrimidin-4-amine |
11222252 |
ChemBL |
YES1 |
HGNC:12841 |
P07947 |
N-(2-methoxyphenyl)-5-phenyl-1,3-oxazol-2-amine;hydrochloride |
11231939 |
DSigDB |
YES1 |
HGNC:12841 |
P07947 |
4-(4-fluorophenyl)-N-(1H-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide |
11233873 |
DGidb |
YES1 |
HGNC:12841 |
P07947 |
Brivanib |
11234052 |
DSigDB |
YES1 |
HGNC:12841 |
P07947 |
3-(4-Amino-3-(3-chloro-4-fluorophenyl)thieno[3,2-c]pyridin-7-yl)benzenesulfonamide |
11281930 |
DGidb |