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Drugs And Genes
DRUGs and GENEs
GENE_SYMBOL HGNC_ID UNIPROT_ID DRUG_NAME PUBCHEM_CID Datasource
ADORA2B HGNC:264 P29275 (2R,3R,4S,5R)-2-[6-(cyclopentylamino)-2-(3,5-dimethylphenyl)purin-9-yl]-5-[(3,5-dimethylpyrazol-1-yl)methyl]oxolane-3,4-diol 137651531 BindingDB
ADORA2B HGNC:264 P29275 (2R,3R,4S,5R)-2-[2-chloro-6-(4-chloro-2-fluoroanilino)purin-9-yl]-5-[(3,5-dimethylpyrazol-1-yl)methyl]oxolane-3,4-diol 137652383 BindingDB
ADORA2B HGNC:264 P29275 (2R,3R,4S,5R)-2-[6-(2-bicyclo[2.2.1]heptanylamino)purin-9-yl]-5-[(3,5-dimethylpyrazol-1-yl)methyl]oxolane-3,4-diol 137653588 BindingDB
ADORA2B HGNC:264 P29275 (2R,3S,4R,5R)-2-[(3,5-dimethylpyrazol-1-yl)methyl]-5-[6-[[(3R)-oxolan-3-yl]amino]purin-9-yl]oxolane-3,4-diol 137656139 BindingDB
ADORA2B HGNC:264 P29275 (2R,3R,4S,5R)-2-[6-(4-chloro-2-fluoroanilino)-2-(3,5-dimethylphenyl)purin-9-yl]-5-[(3,5-dimethylpyrazol-1-yl)methyl]oxolane-3,4-diol 137657382 BindingDB
ADORA2B HGNC:264 P29275 (2R,3R,4S,5R)-2-[6-(4-chloro-2-fluoroanilino)purin-9-yl]-5-[(3,5-dimethylpyrazol-1-yl)methyl]oxolane-3,4-diol 137657570 BindingDB
ADORA2B HGNC:264 P29275 (2R,3R,4S,5R)-2-[6-(2-bicyclo[2.2.1]heptanylamino)-2-(3,5-dimethylphenyl)purin-9-yl]-5-[(3,5-dimethylpyrazol-1-yl)methyl]oxolane-3,4-diol 137661322 BindingDB
ADORA2B HGNC:264 P29275 (2R,3R,4S,5R)-2-[2-chloro-6-[(4-chloro-2-fluorophenyl)methylamino]purin-9-yl]-5-(2-ethyltetrazol-5-yl)oxolane-3,4-diol 137661670 BindingDB
ADORA2B HGNC:264 P29275 4-hydroxy-N-(4-methoxy-7-morpholin-4-yl-1,3-benzothiazol-2-yl)-1-methylcyclohexane-1-carboxamide 137661874 BindingDB
ADORA2B HGNC:264 P29275 Methyl 3-[[6-amino-3,5-dicyano-4-(furan-2-yl)pyridin-2-yl]sulfanylmethyl]benzoate 139030524 BindingDB
ADORA2B HGNC:264 P29275 US11168089, Ex. No. 3 139508736 BindingDB
ADORA2B HGNC:264 P29275 7,8-Dihydroxy-3-(4-hydroxyphenyl)chromen-2-one 141536950 BindingDB
ADORA2B HGNC:264 P29275 N-[(3R)-1-[2-[[(1S)-1-pyridin-2-ylethyl]amino]thieno[3,2-d]pyrimidine-4-carbonyl]pyrrolidin-3-yl]acetamide 142540040 BindingDB
ADORA2B HGNC:264 P29275 N-[(2R)-2-hydroxypropyl]-6-methyl-2-[[(1S)-1-pyridin-3-ylethyl]amino]thieno[3,2-d]pyrimidine-4-carboxamide 142540051 BindingDB
ADORA2B HGNC:264 P29275 1-[3-[2-[[(1S)-1-(5-fluoropyridin-3-yl)ethyl]amino]thieno[3,2-d]pyrimidine-4-carbonyl]imidazolidin-1-yl]-2,2-dimethylpropan-1-one 142540081 BindingDB
ADORA2B HGNC:264 P29275 [2-[[(1S)-1-(5-fluoropyridin-3-yl)ethyl]amino]-6-methylthieno[3,2-d]pyrimidin-4-yl]-[(3R)-3-hydroxypyrrolidin-1-yl]methanone 142540095 BindingDB
ADORA2B HGNC:264 P29275 azetidin-1-yl-[2-[[(1S)-1-(5-fluoropyridin-3-yl)ethyl]amino]thieno[3,2-d]pyrimidin-4-yl]methanone 142540098 BindingDB
ADORA2B HGNC:264 P29275 [2-[[(1S)-1-(5-fluoropyridin-3-yl)ethyl]amino]-6-(trifluoromethyl)thieno[3,2-d]pyrimidin-4-yl]-[(3R)-3-hydroxypyrrolidin-1-yl]methanone 142540105 BindingDB
ADORA2B HGNC:264 P29275 N-[1-[2-[[(1S)-1-(5-fluoropyridin-3-yl)ethyl]amino]thieno[3,2-d]pyrimidine-4-carbonyl]azetidin-3-yl]oxolane-3-carboxamide 142540138 BindingDB
ADORA2B HGNC:264 P29275 [(3R)-3-hydroxypyrrolidin-1-yl]-[6-methyl-2-[[(1S)-1-pyridin-2-ylethyl]amino]thieno[3,2-d]pyrimidin-4-yl]methanone 142540146 BindingDB