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Drugs And Genes
DRUGs and GENEs
GENE_SYMBOL HGNC_ID UNIPROT_ID DRUG_NAME PUBCHEM_CID Datasource
ADORA3 HGNC:268 P0DMS8 [(3S)-3-hydroxypyrrolidin-1-yl]-[6-methyl-2-[[(1S)-1-pyridin-3-ylethyl]amino]thieno[3,2-d]pyrimidin-4-yl]methanone 153637795 BindingDB
ADORA3 HGNC:268 P0DMS8 (3-methoxyazetidin-1-yl)-[2-[[(1S)-1-pyridin-3-ylethyl]amino]thieno[3,2-d]pyrimidin-4-yl]methanone 153637796 BindingDB
ADORA3 HGNC:268 P0DMS8 (3-hydroxyazetidin-1-yl)-[2-[[(1S)-1-pyridin-3-ylethyl]amino]thieno[3,2-d]pyrimidin-4-yl]methanone 153637799 BindingDB
ADORA3 HGNC:268 P0DMS8 2-[[(1S)-1-(5-fluoropyridin-3-yl)ethyl]amino]-N-[(2R)-2-hydroxypropyl]thieno[3,2-d]pyrimidine-4-carboxamide 153637803 BindingDB
ADORA3 HGNC:268 P0DMS8 [2-[[(1S)-1-(5-fluoropyridin-3-yl)ethyl]amino]-6-methylthieno[3,2-d]pyrimidin-4-yl]-[(3R)-3-(hydroxymethyl)pyrrolidin-1-yl]methanone 153637804 BindingDB
ADORA3 HGNC:268 P0DMS8 [2-[[(1S)-1-(5-fluoropyridin-3-yl)ethyl]amino]thieno[3,2-d]pyrimidin-4-yl]-[(3S)-3-hydroxypyrrolidin-1-yl]methanone 153637805 BindingDB
ADORA3 HGNC:268 P0DMS8 [(3S)-3-(methoxymethyl)pyrrolidin-1-yl]-[6-methyl-2-[[(1S)-1-pyridin-2-ylethyl]amino]thieno[3,2-d]pyrimidin-4-yl]methanone 153637814 BindingDB
ADORA3 HGNC:268 P0DMS8 [(3S)-3-(hydroxymethyl)pyrrolidin-1-yl]-[2-[[(1S)-1-pyridin-3-ylethyl]amino]thieno[3,2-d]pyrimidin-4-yl]methanone 153637815 BindingDB
ADORA3 HGNC:268 P0DMS8 [(3R)-3-(aminomethyl)pyrrolidin-1-yl]-[2-[[(1S)-1-(5-fluoropyridin-3-yl)ethyl]amino]-6-methylthieno[3,2-d]pyrimidin-4-yl]methanone 153637817 BindingDB
ADORA3 HGNC:268 P0DMS8 (3-aminoazetidin-1-yl)-[2-[[(1S)-1-(5-fluoropyridin-3-yl)ethyl]amino]-6-methylthieno[3,2-d]pyrimidin-4-yl]methanone 153637818 BindingDB
ADORA3 HGNC:268 P0DMS8 N-[(3S)-1-[2-[(5-fluoropyridin-3-yl)methylamino]thieno[3,2-d]pyrimidine-4-carbonyl]pyrrolidin-3-yl]-2,2-dimethylpropanamide 153637820 BindingDB
ADORA3 HGNC:268 P0DMS8 [(3S)-3-(hydroxymethyl)pyrrolidin-1-yl]-[6-methyl-2-[[(1S)-1-pyridin-3-ylethyl]amino]thieno[3,2-d]pyrimidin-4-yl]methanone 153637826 BindingDB
ADORA3 HGNC:268 P0DMS8 [(3S)-3-methylpyrrolidin-1-yl]-[2-[[(1S)-1-pyridin-2-ylethyl]amino]thieno[3,2-d]pyrimidin-4-yl]methanone 153637835 BindingDB
ADORA3 HGNC:268 P0DMS8 [6-amino-2-[[(1S)-1-(5-fluoropyridin-3-yl)ethyl]amino]thieno[3,2-d]pyrimidin-4-yl]-[(3R)-3-hydroxypyrrolidin-1-yl]methanone 153637836 BindingDB
ADORA3 HGNC:268 P0DMS8 [2-[[(1S)-1-(5-fluoropyridin-3-yl)ethyl]amino]-6-methylthieno[3,2-d]pyrimidin-4-yl]-[(2R)-2-methylazetidin-1-yl]methanone 153637837 BindingDB
ADORA3 HGNC:268 P0DMS8 benzyl N-[(3R)-1-[2-[[(1S)-1-(5-fluoropyridin-3-yl)ethyl]amino]-6-methylthieno[3,2-d]pyrimidine-4-carbonyl]pyrrolidin-3-yl]carbamate 153637838 BindingDB
ADORA3 HGNC:268 P0DMS8 [6-amino-2-[[(1S)-1-(5-fluoropyridin-3-yl)ethyl]amino]thieno[3,2-d]pyrimidin-4-yl]-(azetidin-1-yl)methanone 153637843 BindingDB
ADORA3 HGNC:268 P0DMS8 [2-[[(1S)-1-(5-fluoropyridin-3-yl)ethyl]amino]thieno[3,2-d]pyrimidin-4-yl]-[(3R)-3-(hydroxymethyl)pyrrolidin-1-yl]methanone 153637846 BindingDB
ADORA3 HGNC:268 P0DMS8 [(3R)-3-aminopyrrolidin-1-yl]-[2-[[(1S)-1-(5-fluoropyridin-3-yl)ethyl]amino]-6-methylthieno[3,2-d]pyrimidin-4-yl]methanone 153637847 BindingDB
ADORA3 HGNC:268 P0DMS8 N-[[1-[2-[[(1S)-1-(5-fluoropyridin-3-yl)ethyl]amino]thieno[3,2-d]pyrimidine-4-carbonyl]azetidin-3-yl]methyl]-2-methylpropanamide 153637849 BindingDB