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Drugs And Genes
DRUGs and GENEs
GENE_SYMBOL HGNC_ID UNIPROT_ID DRUG_NAME PUBCHEM_CID Datasource
ADORA3 HGNC:268 P0DMS8 (1S,2R,3S,4R,5S)-4-[5-chloro-7-(ethylamino)imidazo[4,5-b]pyridin-3-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 162735387 BindingDB
ADORA3 HGNC:268 P0DMS8 (1S,2R,3S,4R,5S)-4-[5-chloro-7-[[5-chloro-2-[(3-methyl-1,2-oxazol-5-yl)methoxy]phenyl]methylamino]imidazo[4,5-b]pyridin-3-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 162735491 BindingDB
ADORA3 HGNC:268 P0DMS8 (1R,2R,3S,4R,5S)-4-[2-chloro-6-(2,2-difluoroethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol 162735527 BindingDB
ADORA3 HGNC:268 P0DMS8 N-(3-hydroxycyclobutyl)-2-[[(1S)-1-pyridin-2-ylethyl]amino]thieno[3,2-d]pyrimidine-4-carboxamide 162779409 BindingDB
ADORA3 HGNC:268 P0DMS8 2-[[(1S)-1-(5-chloropyridin-3-yl)ethyl]amino]-N-(3-hydroxycyclobutyl)thieno[3,2-d]pyrimidine-4-carboxamide 162779426 BindingDB
ADORA3 HGNC:268 P0DMS8 N-(2,2-dimethylpropyl)-1-[2-[[(1S)-1-(5-fluoropyridin-3-yl)ethyl]amino]thieno[3,2-d]pyrimidine-4-carbonyl]pyrrolidine-3-carboxamide 162779488 BindingDB
ADORA3 HGNC:268 P0DMS8 4-[2-[7-amino-4-(furan-2-yl)-3,5,6,8,10,11-hexazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7,11-pentaen-10-yl]ethyl]-N-(2-aminophenyl)benzamide 163196437 BindingDB
ADORA3 HGNC:268 P0DMS8 (3-hydroxypyrrolidin-1-yl)-[6-(methylamino)-2-[[(1S)-1-pyridin-3-ylethyl]amino]thieno[3,2-d]pyrimidin-4-yl]methanone 163408067 BindingDB
ADORA3 HGNC:268 P0DMS8 N-[(3R)-3-hydroxycyclopentyl]-2-[[(1S)-1-pyridin-2-ylethyl]amino]thieno[3,2-d]pyrimidine-4-carboxamide 163408070 BindingDB
ADORA3 HGNC:268 P0DMS8 NMDA receptor modulator 3 163408779 BindingDB
ADORA3 HGNC:268 P0DMS8 (2R,3R,4S,5R)-2-[2-chloro-6-(4-phenylbutylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol 164619608 BindingDB
ADORA3 HGNC:268 P0DMS8 A2Aar/hdac-IN-1 165412579 BindingDB
ADORA3 HGNC:268 P0DMS8 A2Aar/hdac-IN-2 165412580 BindingDB
ADORA3 HGNC:268 P0DMS8 4-[4-(3-piperidin-1-ylpropoxy)phenyl]-5H-indeno[1,2-d]pyrimidin-2-amine 166631046 BindingDB
ADORA3 HGNC:268 P0DMS8 (2E)-1-[6-[[3-[[3-[2-[[4-(2,6-dioxo-1,3-dipropyl-7H-purin-8-yl)bicyclo[2.2.2]octane-1-carbonyl]amino]ethylamino]-3-oxopropyl]amino]-3-oxopropyl]amino]-6-oxohexyl]-3,3-dimethyl-2-[(2E,4E)-5-(1,3,3-trimethyl-5-sulfoindol-1-ium-2-yl)penta-2,4-dienylidene]indole-5-sulfonate 166631966 BindingDB
ADORA3 HGNC:268 P0DMS8 2-Amino-4-[4-(3-piperidin-1-ylpropoxy)phenyl]indeno[1,2-d]pyrimidin-5-one 166632350 BindingDB
ADORA3 HGNC:268 P0DMS8 7-(3-piperidin-1-ylpropoxy)-4-[4-(3-piperidin-1-ylpropoxy)phenyl]-5H-indeno[1,2-d]pyrimidin-2-amine 166633096 BindingDB
ADORA3 HGNC:268 P0DMS8 4-phenyl-7-(3-piperidin-1-ylpropoxy)-5H-indeno[1,2-d]pyrimidin-2-amine 166633426 BindingDB
ADORA3 HGNC:268 P0DMS8 4-phenyl-7-(3-pyrrolidin-1-ylpropoxy)-5H-indeno[1,2-d]pyrimidin-2-amine 166635863 BindingDB
ADORA3 HGNC:268 P0DMS8 2-Amino-4-phenyl-7-(3-piperidin-1-ylpropoxy)indeno[1,2-d]pyrimidin-5-one 166635957 BindingDB