| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| AKT3 |
HGNC:393 |
Q9Y243 |
(13r,15s)-13-Methyl-16-Oxa-8,9,12,22,24-Pentaazahexacyclo[15.6.2.16,9.1,12,15.0,2,7.0,21,25]heptacosa-1(24),2,4,6,17(25),18,20-Heptaene-23,26-Dione |
16046126 |
BindingDB |
| AKT3 |
HGNC:393 |
Q9Y243 |
Fedratinib |
16722836 |
BindingDB |
| AKT3 |
HGNC:393 |
Q9Y243 |
Pictilisib |
17755052 |
BindingDB |
| AKT3 |
HGNC:393 |
Q9Y243 |
1-(1-{[4-(3-phenylquinolin-2-yl)phenyl]methyl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one |
21103107 |
BindingDB |
| AKT3 |
HGNC:393 |
Q9Y243 |
1-[1-({4-[6-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-3-phenylquinoxalin-2-yl]phenyl}methyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one |
21103111 |
BindingDB |
| AKT3 |
HGNC:393 |
Q9Y243 |
1-[1-({4-[7-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-3-phenylquinoxalin-2-yl]phenyl}methyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one |
21103119 |
BindingDB |
| AKT3 |
HGNC:393 |
Q9Y243 |
2-(4-{[4-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]methyl}phenyl)-3-phenylquinoxaline-6-carboxylic acid |
21103197 |
BindingDB |
| AKT3 |
HGNC:393 |
Q9Y243 |
1-(1-{[4-(6-benzyl-5-oxo-3-phenyl-4,5-dihydropyrazin-2-yl)phenyl]methyl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one |
23647016 |
BindingDB |
| AKT3 |
HGNC:393 |
Q9Y243 |
1-{1-[(4-{6-[(4-hydroxyphenyl)methyl]-5-oxo-3-phenyl-4,5-dihydropyrazin-2-yl}phenyl)methyl]piperidin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one |
23647018 |
BindingDB |
| AKT3 |
HGNC:393 |
Q9Y243 |
1-{1-[(4-{5-[(4-hydroxyphenyl)methyl]-6-oxo-3-phenyl-1,6-dihydropyrazin-2-yl}phenyl)methyl]piperidin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one |
23647019 |
BindingDB |
| AKT3 |
HGNC:393 |
Q9Y243 |
1-(1-{[4-(2-phenylquinolin-3-yl)phenyl]methyl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one |
23647020 |
BindingDB |
| AKT3 |
HGNC:393 |
Q9Y243 |
N-(3-(5-chloro-1H-pyrrolo[2,3-b]pyridine-3-carbonyl)-2,4-difluorophenyl)propane-1-sulfonamide |
24180719 |
BindingDB |
| AKT3 |
HGNC:393 |
Q9Y243 |
4-[6-[4-(2-piperidin-1-ylethoxy)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]-N-(2,2,2-trifluoroethyl)thiophene-2-carboxamide |
24759534 |
BindingDB |
| AKT3 |
HGNC:393 |
Q9Y243 |
(2S)-2-(4-chlorophenyl)-1-[4-[(5R,7R)-7-fluoro-5-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl]piperazin-1-yl]-3-(propan-2-ylamino)propan-1-one |
24783593 |
BindingDB |
| AKT3 |
HGNC:393 |
Q9Y243 |
(2S)-2-(4-chlorophenyl)-3-(4-fluoropiperidin-1-yl)-1-[4-[(5R,7R)-7-hydroxy-5-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl]piperazin-1-yl]propan-1-one |
24788164 |
BindingDB |
| AKT3 |
HGNC:393 |
Q9Y243 |
Quizartinib |
24889392 |
BindingDB |
| AKT3 |
HGNC:393 |
Q9Y243 |
Ruxolitinib |
25126798 |
BindingDB |
| AKT3 |
HGNC:393 |
Q9Y243 |
2-((2-((1-(2-(Dimethylamino)acetyl)-5-methoxyindolin-6-yl)amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino)-6-fluoro-N-methylbenzamide |
25182616 |
BindingDB |
| AKT3 |
HGNC:393 |
Q9Y243 |
6-{[(2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihydroxyoxolan-2-yl]formamido}hexanamide |
25190765 |
BindingDB |
| AKT3 |
HGNC:393 |
Q9Y243 |
3-(3-Iodobenzyl)-1-tert-butyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine |
25243798 |
BindingDB |