GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
ABL1 |
HGNC:76 |
P00519 |
6-(2,6-dichlorophenyl)-8-methyl-2-(4-(3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yloxy)phenylamino)pyrido[2,3-d]pyrimidin-7(8H)-one |
45487997 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
Larotrectinib |
46188928 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
Pha-793887 |
46191454 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
Bemcentinib |
46215462 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
5-(2-aminoethyl)-7-(7-(benzo[b]thiophen-2-yl)-1H-indazol-5-yl)-5H-pyrrolo[3,2-d]pyrimidin-2-amine |
46224684 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
4-amino-5-(2,6-difluorobenzoyl)-2-(4-phenoxyphenyl)-1H-pyrrole-3-carboxamide |
46224908 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
(R)-6-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)quinoline |
46232443 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
(R)-3-(6-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)quinolin-3-yl)acrylamide |
46232555 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
2-(6-((R)-1-(2,6-dichloro-3-fluorophenyl)ethoxy)quinolin-3-yl)cyclopropanecarboxamide |
46232556 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
3-((4-(Dimethylamino)naphthalen-1-yl)methylene)-4-methylindolin-2-one |
46233185 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
N,1-dimethyl-8-[[1-(1-methylsulfonylpiperidine-4-carbonyl)piperidin-4-yl]amino]-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide |
46233287 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
3-(Naphthalen-1-Ylmethyl)-1-(Piperidin-4-Ylmethyl)-1h-Pyrazolo[3,4-D]pyrimidin-4-Amine |
46398830 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
2-(6-(4-(Trifluoromethoxy)phenylamino)pyrimidin-4-yl)benzamide |
46703970 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
2-[(2-Oxo-2-phenylethyl)sulfanyl]-4-(3-thienyl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile |
46838818 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
Flumatinib |
46848036 |
BindingDB, TTD |
ABL1 |
HGNC:76 |
P00519 |
5-[(2-bromobenzoyl)amino]-N-[3-(dimethylamino)propyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxamide |
46861577 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
5-((5-(4-((4-(2-hydroxyethyl)piperazin-1-yl)methyl)-3-(trifluoromethyl)phenylcarbamoyl)-2-methylphenyl)ethynyl)-N,1-dimethyl-1H-imidazole-2-carboxamide |
46864270 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
(E)-2-(4-Bromobenzylthio)-3-(4-fluoro-3-nitrophenyl)-1-(4-(4-(2-hydroxy-ethyl)piperazine-1-carbonyl)phenyl)prop-2-en-1-one |
46865999 |
TTD |
ABL1 |
HGNC:76 |
P00519 |
(E)-3-(4-Fluoro-3-nitrophenyl)-2-(4-fluorobenzylthio)-1-(4-(4-(2-hydroxyethyl)piperazine-1-carbonyl)phenyl)prop-2-en-1-one |
46866098 |
TTD |
ABL1 |
HGNC:76 |
P00519 |
(E)-4-(3-(4-Fluoro-3-nitrophenyl)-2-(4-(trifluoromethyl)benzylthio)acryloyl)benzoic acid |
46866099 |
TTD |