| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| ACVR1 |
HGNC:171 |
Q04771 |
3-[4-[3-(2-Methylquinolin-4-yl)imidazo[1,2-a]pyridin-7-yl]phenyl]morpholine |
139495370 |
BindingDB |
| ACVR1 |
HGNC:171 |
Q04771 |
3-[4-[3-(6-Fluoro-2-methylquinolin-4-yl)imidazo[1,2-a]pyridin-7-yl]phenyl]morpholine |
139495455 |
BindingDB |
| ACVR1 |
HGNC:171 |
Q04771 |
2-Methyl-4-[7-(4-piperazin-2-ylphenyl)imidazo[1,2-a]pyridin-3-yl]quinoline |
139495458 |
BindingDB |
| ACVR1 |
HGNC:171 |
Q04771 |
6-Methoxy-4-[6-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-3-yl]quinolin-7-ol |
142464127 |
BindingDB |
| ACVR1 |
HGNC:171 |
Q04771 |
6-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]-4-(oxan-4-yloxy)-3-(1H-pyrazol-4-yl)pyrazolo[1,5-a]pyridine |
142464133 |
BindingDB |
| ACVR1 |
HGNC:171 |
Q04771 |
7-Fluoro-6-methoxy-4-[7-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]imidazo[1,2-a]pyridin-3-yl]quinoline |
142464146 |
BindingDB |
| ACVR1 |
HGNC:171 |
Q04771 |
8-Fluoro-6-methoxy-4-[6-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-3-yl]quinoline |
142464149 |
BindingDB |
| ACVR1 |
HGNC:171 |
Q04771 |
4-[6-[4-(4,4-Dimethylpiperazin-4-ium-1-yl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-3-yl]-7-fluoro-6-methoxyquinoline |
142464157 |
BindingDB |
| ACVR1 |
HGNC:171 |
Q04771 |
3-(7-Fluoro-6-methoxyquinolin-4-yl)-6-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-2-amine |
142464171 |
BindingDB |
| ACVR1 |
HGNC:171 |
Q04771 |
N-methyl-4-[6-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-2-carboxamide |
142464174 |
BindingDB |
| ACVR1 |
HGNC:171 |
Q04771 |
6-[3-(4-Methylpiperazin-1-yl)azetidin-1-yl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine |
142464194 |
BindingDB |
| ACVR1 |
HGNC:171 |
Q04771 |
4-[6-[4-(4-Methylpiperazin-1-yl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-3-yl]-6-(trifluoromethoxy)quinoline |
142464200 |
BindingDB |
| ACVR1 |
HGNC:171 |
Q04771 |
1-[3-(7-Fluoro-6-methoxyquinolin-4-yl)pyrazolo[1,5-a]pyrimidin-6-yl]piperazin-2-one |
142464210 |
BindingDB |
| ACVR1 |
HGNC:171 |
Q04771 |
6-Methyl-4-[6-[3-(4-methylpiperazin-1-yl)azetidin-1-yl]pyrazolo[1,5-a]pyrimidin-3-yl]quinoline |
142464217 |
BindingDB |
| ACVR1 |
HGNC:171 |
Q04771 |
1-[4-[4-(3-Quinolin-4-ylpyrazolo[1,5-a]pyrimidin-6-yl)piperazin-1-yl]piperidin-1-yl]ethanone |
142464239 |
BindingDB |
| ACVR1 |
HGNC:171 |
Q04771 |
6-[4-(4-Methylpiperazin-1-yl)piperidin-1-yl]-3-(1-methylpyrrolo[2,3-b]pyridin-4-yl)pyrazolo[1,5-a]pyrimidine |
142464268 |
BindingDB |
| ACVR1 |
HGNC:171 |
Q04771 |
7-Fluoro-6-methoxy-4-[6-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]-4-(oxan-4-yloxy)pyrazolo[1,5-a]pyridin-3-yl]quinoline |
142464278 |
BindingDB |
| ACVR1 |
HGNC:171 |
Q04771 |
5-Fluoro-6-methyl-4-[6-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-3-yl]quinoline |
142464282 |
BindingDB |
| ACVR1 |
HGNC:171 |
Q04771 |
7-Fluoro-4-[6-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-3-yl]quinolin-6-ol |
142464328 |
BindingDB |
| ACVR1 |
HGNC:171 |
Q04771 |
2-Methyl-4-[6-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-3-yl]-7-(trifluoromethyl)quinoline |
142464333 |
BindingDB |