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Drugs And Genes
DRUGs and GENEs
GENE_SYMBOL HGNC_ID UNIPROT_ID DRUG_NAME PUBCHEM_CID Datasource
ACVR1 HGNC:171 Q04771 ((2S)-1-(1-(tetrahydro-2H-pyran-2-yl)-4-((1-(3,4,5-trimethoxyphenyl)-1H-imidazol-4-yl)amino)-1H-pyrazolo[3,4-d]pyrimidin-6-yl)pyrrolidin-2-yl)methanol 142498181 BindingDB
ACVR1 HGNC:171 Q04771 (S)-(1-(4-((1-(3-bromo-4-(trifluoromethoxy)phenyl)-1H-imidazol-4-yl)amino)pyrrolo[2,1-f][1,2,4]triazin-2-yl)pyrrolidin-2-yl)methanol 142498184 BindingDB
ACVR1 HGNC:171 Q04771 (S)-(1-(4-chloroquinolin-2-yl)pyrrolidin-2-yl)methanol 142498193 BindingDB
ACVR1 HGNC:171 Q04771 (S)-(1-(8-isopropoxy-4-((1-(3,4,5-trimethoxyphenyl)-1H-imidazol-4-yl)amino)quinazolin-2-yl)pyrrolidin-2-yl)methanol 142498197 BindingDB
ACVR1 HGNC:171 Q04771 N-(1-methyl-1H-imidazol-4-yl)-2-(2-(pyridin-2-yl)pyrrolidin-1-yl)furo[3,2-d]pyrimidin-4-amine 142498200 BindingDB
ACVR1 HGNC:171 Q04771 (R)-(1-(2-(1-(3,4,5-trimethoxyphenyl)-1H-imidazol-4-ylamino)-6,7-dihydro-5H-pyrrolo[3,4-d]pyrimidin-4-yl)pyrrolidin-2-yl)methanol 142498202 BindingDB
ACVR1 HGNC:171 Q04771 3-(6-(hydroxymethyl)-4-((1-(3,4,5-trimethoxyphenyl)-1H-imidazol-4-yl)amino)thieno[2,3-d]pyrimidin-2-yl)benzaldehyde 142498207 BindingDB
ACVR1 HGNC:171 Q04771 (3-(6-(hydroxymethyl)-4-((1-(3,4,5-trimethoxyphenyl)-1H-imidazol-4-yl)amino)thieno[2,3-d]pyrimidin-2-yl)phenyl)methanol 142498208 BindingDB
ACVR1 HGNC:171 Q04771 N2,N7-bis(1-(3,4,5-trimethoxyphenyl)-1H-imidazol-4-yl)naphthalene-2,7-diamine 142498211 BindingDB
ACVR1 HGNC:171 Q04771 (S)-2-(4-(2-(hydroxymethyl)pyrrolidin-1-yl)-2-((1-(3,4,5-trimethoxyphenyl)-1H-imidazol-4-yl)amino)-5,6-dihydropyrido[3,4-d]pyrimidin-7(8H)-yl)acetamide 142498214 BindingDB
ACVR1 HGNC:171 Q04771 (S)-(1-(2-((1-(3,4,5-trimethoxyphenyl)-1H-imidazol-4-yl)amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-2-yl)methanol 142498216 BindingDB
ACVR1 HGNC:171 Q04771 (S)-N-(3-(4-(2-(hydroxymethyl)pyrrolidin-1-yl)-2-((1-(3,4,5-trimethoxyphenyl)-1H-imidazol-4-yl)amino)quinazolin-7-yl)phenyl)acetamide 142498223 BindingDB
ACVR1 HGNC:171 Q04771 (S)-1-(4-(1-(3,4,5-trimethoxyphenyl)-1H-imidazol-4-ylamino)pyrrolo[2,1-f][1,2,4]triazin-2-yl)pyrrolidine-2-carboxamide 142498232 BindingDB
ACVR1 HGNC:171 Q04771 (S)-2-(3-(dimethylamino)pyrrolidin-1-yl)-N-(1-(3,4,5-trimethoxyphenyl)-1H-imidazol-4-yl)furo[3,2-d]pyrimidin-4-amine 142498238 BindingDB
ACVR1 HGNC:171 Q04771 (cis)-3-(4-((S)-2-(hydroxymethyl)pyrrolidin-1-yl)-3-methyl-6-((1-(3,4,5-trimethoxyphenyl)-1H-imidazol-4-yl)amino)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)cyclobutanol 142498239 BindingDB
ACVR1 HGNC:171 Q04771 (R)-(1-(2-((1-(3,4,5-trimethoxyphenyl)-1H-imidazol-4-yl)amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-2-yl)methanol 142498241 BindingDB
ACVR1 HGNC:171 Q04771 (S)-(1-(2-((1-(3-methyl-5-(trifluoromethoxy)phenyl)-1H-imidazol-4-yl)amino)pyrrolo[2,1-f][1,2,4]triazin-4-yl)pyrrolidin-2-yl)methanol 142498242 BindingDB
ACVR1 HGNC:171 Q04771 (S)-(1-(4-((1-(3,4,5-trimethoxyphenyl)-1H-imidazol-4-yl)amino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidin-2-yl)methanol 142498244 BindingDB
ACVR1 HGNC:171 Q04771 (S)-(1-(7-(3-aminophenyl)-2-((1-(3,4,5-trimethoxyphenyl)-1H-imidazol-4-yl)amino)quinazolin-4-yl)pyrrolidin-2-yl)methanol 142498249 BindingDB
ACVR1 HGNC:171 Q04771 (S)-(1-(7-(1,2,3,6-tetrahydropyridin-4-yl)-4-(1-(3,4,5-trimethoxyphenyl)-1H-imidazol-4-ylamino)pyrrolo[2,1-f][1,2,4]triazin-2-yl)pyrrolidin-2-yl)methanol 142498251 BindingDB