| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| WDR5 |
HGNC:12757 |
P61964 |
5-bromo-3-chloro-N-[1-cyclopentyl-2-(methylsulfonyl)-1H-imidazol-4-yl]-2-hydroxybenzene-1-sulfonamide |
146019259 |
ChemBL |
| WDR5 |
HGNC:12757 |
P61964 |
US10807959, Example B5 |
146370875 |
ChemBL |
| WDR5 |
HGNC:12757 |
P61964 |
N-[(4-chloro-3-methylphenyl)methyl]-3-(4-fluoro-2-methylphenyl)-5-[(2-imino-3-methylimidazol-1-yl)methyl]benzamide |
146456000 |
ChemBL |
| WDR5 |
HGNC:12757 |
P61964 |
3-(4-fluoro-2-methylphenyl)-N-[(4-fluoro-3-methylphenyl)methyl]-5-[(2-imino-3-methylimidazol-1-yl)methyl]benzamide |
146456497 |
ChemBL |
| WDR5 |
HGNC:12757 |
P61964 |
7-[(2-Methylimidazol-1-yl)methyl]-2-[(2-methylpyridin-4-yl)methyl]-5-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]-3,4-dihydroisoquinolin-1-one |
147934765 |
ChemBL |
| WDR5 |
HGNC:12757 |
P61964 |
7-[(2-Methylimidazol-1-yl)methyl]-5-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]-2-(pyridin-2-ylmethyl)-3,4-dihydroisoquinolin-1-one |
153238800 |
ChemBL |
| WDR5 |
HGNC:12757 |
P61964 |
N-[5-[2-fluoro-5-[[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethyl]carbamoyl]phenyl]-2-[(3R,5S)-3,4,5-trimethylpiperazin-1-yl]phenyl]-6-oxo-4-(trifluoromethyl)-1H-pyridine-3-carboxamide |
153379991 |
GtoPDB |
| WDR5 |
HGNC:12757 |
P61964 |
WDR5 degrader MS40 |
153380106 |
GtoPDB |
| WDR5 |
HGNC:12757 |
P61964 |
2-[(3,5-Dimethoxyphenyl)methyl]-5-(1,3-dimethylpyrazol-4-yl)-7-[(2-imino-3-methylimidazol-1-yl)methyl]-3,4-dihydroisoquinolin-1-one |
153572276 |
ChemBL |
| WDR5 |
HGNC:12757 |
P61964 |
7-[(2-Methylimidazol-1-yl)methyl]-2-[(4-methylpyridin-2-yl)methyl]-5-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]-3,4-dihydroisoquinolin-1-one |
153572325 |
ChemBL |
| WDR5 |
HGNC:12757 |
P61964 |
2-[(3,5-Dimethoxyphenyl)methyl]-5-(4-fluoro-2-methylphenyl)-7-[(5-imino-1-methyl-1,2,4-triazol-4-yl)methyl]-3,4-dihydroisoquinolin-1-one |
153572410 |
ChemBL |
| WDR5 |
HGNC:12757 |
P61964 |
2-[(3,5-Dimethoxyphenyl)methyl]-5-(4-fluoro-2-methylphenyl)-7-[(2-iminopyrrolidin-1-yl)methyl]-3,4-dihydroisoquinolin-1-one |
153572445 |
ChemBL |
| WDR5 |
HGNC:12757 |
P61964 |
2-[(3,5-Dimethoxyphenyl)methyl]-5-(4-fluoro-2-methylphenyl)-7-[(2-imino-1,3-thiazolidin-3-yl)methyl]-3,4-dihydroisoquinolin-1-one |
153572528 |
ChemBL |
| WDR5 |
HGNC:12757 |
P61964 |
2-[(3,5-Dimethoxyphenyl)methyl]-7-[(2-imino-3-methylimidazol-1-yl)methyl]-5-(1,3,5-trimethylpyrazol-4-yl)-3,4-dihydroisoquinolin-1-one |
153572559 |
ChemBL |
| WDR5 |
HGNC:12757 |
P61964 |
7-[(2-Methylimidazol-1-yl)methyl]-2-[(3-methylpyridin-2-yl)methyl]-5-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]-3,4-dihydroisoquinolin-1-one |
153572565 |
ChemBL |
| WDR5 |
HGNC:12757 |
P61964 |
7-[(3-Cyclopropyl-2-iminoimidazol-1-yl)methyl]-2-[(3,5-dimethoxyphenyl)methyl]-5-(4-fluoro-2-methylphenyl)-3,4-dihydroisoquinolin-1-one |
153572603 |
ChemBL |
| WDR5 |
HGNC:12757 |
P61964 |
N'-[[2-[(3,5-dimethoxyphenyl)methyl]-5-(4-fluoro-2-methylphenyl)-1-oxo-3,4-dihydroisoquinolin-7-yl]methyl]cyclopropanecarboximidamide |
153572609 |
ChemBL |
| WDR5 |
HGNC:12757 |
P61964 |
2-[(4-Chloro-3-methylphenyl)methyl]-5-(4-fluoro-2-methylphenyl)-7-[(2-imino-3-methylimidazol-1-yl)methyl]-3,4-dihydroisoquinolin-1-one |
153572631 |
ChemBL |
| WDR5 |
HGNC:12757 |
P61964 |
Wdr5-IN-5 |
153572662 |
GtoPDB |
| WDR5 |
HGNC:12757 |
P61964 |
5-bromo-N-[5-(1-cyanocyclopentyl)-2-hydroxyphenyl]-2-hydroxybenzenesulfonamide |
155511088 |
ChemBL |