| GENE_SYMBOL | 
                HGNC_ID | 
                UNIPROT_ID | 
                DRUG_NAME | 
                PUBCHEM_CID | 
                Datasource | 
            
                                                
                        
                        | YES1 | 
                        HGNC:12841 | 
                        P07947 | 
                        2-(4-(2-(1H-imidazol-1-yl)ethoxy)phenyl)-4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridine | 
                        10294883 | 
                        DGidb | 
                    
                                    
                        
                        | YES1 | 
                        HGNC:12841 | 
                        P07947 | 
                        (R)-6-(4-((4-Ethylpiperazin-1-yl)methyl)phenyl)-N-(1-phenylethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine | 
                        10297043 | 
                        ChemBL, Pubchem, TTD | 
                    
                                    
                        
                        | YES1 | 
                        HGNC:12841 | 
                        P07947 | 
                        N-(5-chloro-2H-1,3-benzodioxol-4-yl)-5-(oxan-4-yloxy)-7-[3-(pyrrolidin-1-yl)propoxy]quinazolin-4-amine | 
                        10301884 | 
                        ChemBL, TTD | 
                    
                                    
                        
                        | YES1 | 
                        HGNC:12841 | 
                        P07947 | 
                        Saracatinib | 
                        10302451 | 
                        ChemBL, DGidb, DSigDB, GtoPDB, Pubchem, TTD | 
                    
                                    
                        
                        | YES1 | 
                        HGNC:12841 | 
                        P07947 | 
                        3-[2-[(Z)-[5-(methylsulfamoyl)-2-oxo-1H-indol-3-ylidene]methyl]-4,5,6,7-tetrahydro-1H-indol-3-yl]propanamide | 
                        10320381 | 
                        ChemBL, TTD | 
                    
                                    
                        
                        | YES1 | 
                        HGNC:12841 | 
                        P07947 | 
                        7-(2,6-dimethylphenyl)-N-phenylbenzo[e][1,2,4]triazin-3-amine | 
                        10404115 | 
                        ChemBL | 
                    
                                    
                        
                        | YES1 | 
                        HGNC:12841 | 
                        P07947 | 
                        5-Ethanesulfonyl-3-[1-{3-[3-(4-methyl-piperazin-1-yl)-propyl]-4,5,6,7-tetrahydro-1H-indol-2-yl}-meth-(Z)-ylidene]-1,3-dihydro-indol-2-one | 
                        10413508 | 
                        ChemBL, TTD | 
                    
                                    
                        
                        | YES1 | 
                        HGNC:12841 | 
                        P07947 | 
                        Tesevatinib | 
                        10458325 | 
                        ChemBL, Pubchem | 
                    
                                    
                        
                        | YES1 | 
                        HGNC:12841 | 
                        P07947 | 
                        [4-(3-{2-[5-Methylsulfamoyl-2-oxo-1,2-dihydro-indol-(3Z)-ylidenemethyl]-4,5,6,7-tetrahydro-1H-indol-3-yl}-propyl)-piperazin-1-yl]-acetic acid | 
                        10482445 | 
                        ChemBL, TTD | 
                    
                                    
                        
                        | YES1 | 
                        HGNC:12841 | 
                        P07947 | 
                        (S)-5-(3-Fluorophenyl)-N-(piperidin-3-yl)-3-ureidothiophene-2-carboxamide | 
                        11152667 | 
                        ChemBL, DGidb, DSigDB, Pubchem | 
                    
                                    
                        
                        | YES1 | 
                        HGNC:12841 | 
                        P07947 | 
                        N-(2-Chloro-6-methylphenyl)-2-((2,6-dimethyl-4-pyrimidinyl)amino)-5-thiazolecarboxamide | 
                        11153014 | 
                        ChemBL, TTD | 
                    
                                    
                        
                        | YES1 | 
                        HGNC:12841 | 
                        P07947 | 
                        5-methyl-7-(3-phenoxyphenyl)-N-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amine | 
                        11155941 | 
                        DGidb | 
                    
                                    
                        
                        | YES1 | 
                        HGNC:12841 | 
                        P07947 | 
                        Sdccggsk-0000152.P001 | 
                        11163861 | 
                        DGidb | 
                    
                                    
                        
                        | YES1 | 
                        HGNC:12841 | 
                        P07947 | 
                        Regorafenib | 
                        11167602 | 
                        DGidb, DSigDB | 
                    
                                    
                        
                        | YES1 | 
                        HGNC:12841 | 
                        P07947 | 
                        Tamatinib | 
                        11213558 | 
                        DGidb, DSigDB | 
                    
                                    
                        
                        | YES1 | 
                        HGNC:12841 | 
                        P07947 | 
                        N-benzyl-1-(2-chloro-2-phenyl-ethyl)pyrazolo[3,4-d]pyrimidin-4-amine | 
                        11222252 | 
                        ChemBL | 
                    
                                    
                        
                        | YES1 | 
                        HGNC:12841 | 
                        P07947 | 
                        N-(2-methoxyphenyl)-5-phenyl-1,3-oxazol-2-amine;hydrochloride | 
                        11231939 | 
                        DSigDB | 
                    
                                    
                        
                        | YES1 | 
                        HGNC:12841 | 
                        P07947 | 
                        4-(4-fluorophenyl)-N-(1H-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide | 
                        11233873 | 
                        DGidb | 
                    
                                    
                        
                        | YES1 | 
                        HGNC:12841 | 
                        P07947 | 
                        Brivanib | 
                        11234052 | 
                        DSigDB | 
                    
                                    
                        
                        | YES1 | 
                        HGNC:12841 | 
                        P07947 | 
                        3-(4-Amino-3-(3-chloro-4-fluorophenyl)thieno[3,2-c]pyridin-7-yl)benzenesulfonamide | 
                        11281930 | 
                        DGidb |