| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| YWHAZ |
HGNC:12855 |
P63104 |
Ac-Gln-Gly-Leu-Leu-Asp-Ala-Leu-Asp-Leu-Ala-Ser-NH2 |
137633432 |
ChemBL |
| YWHAZ |
HGNC:12855 |
P63104 |
(3S)-3-[[(2S)-2-[[(2S,5S,8S,21S)-2-(1-adamantyl)-21-[[2-[[(2S)-5-amino-2-[[2-[2-[2-[(3',6'-dihydroxy-3-oxospiro[2-benzofuran-1,9'-xanthene]-5-yl)carbamothioylamino]ethoxy]ethoxy]acetyl]amino]-5-oxopentanoyl]amino]acetyl]amino]-5-(carboxymethyl)-8,21-dimethyl-3,6,22-trioxo-1,4,7-triazacyclodocosane-8-carbonyl]amino]-4-methylpentanoyl]amino]-4-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-4-oxobutanoic acid |
137635303 |
ChemBL |
| YWHAZ |
HGNC:12855 |
P63104 |
(3S)-3-[[(2S)-2-[[(2S,5S,8S,21S)-21-[[(2R)-2-[[(2S)-5-amino-2-[[2-[2-[2-[(3',6'-dihydroxy-3-oxospiro[2-benzofuran-1,9'-xanthene]-5-yl)carbamothioylamino]ethoxy]ethoxy]acetyl]amino]-5-oxopentanoyl]amino]-3-phenylpropanoyl]amino]-5-(carboxymethyl)-8,21-dimethyl-2-(2-methylpropyl)-3,6,22-trioxo-1,4,7-triazacyclodocosane-8-carbonyl]amino]-4-methylpentanoyl]amino]-4-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-4-oxobutanoic acid |
137635449 |
ChemBL |
| YWHAZ |
HGNC:12855 |
P63104 |
(3S)-3-[[(2S)-2-[[(2S,5S,8S,21S)-21-[[2-[[(2S)-2-acetamido-5-amino-5-oxopentanoyl]amino]acetyl]amino]-5-(carboxymethyl)-8,21-dimethyl-2-(2-methylpropyl)-3,6,22-trioxo-1,4,7-triazacyclodocosane-8-carbonyl]amino]-4-methylpentanoyl]amino]-4-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-4-oxobutanoic acid |
137638149 |
ChemBL |
| YWHAZ |
HGNC:12855 |
P63104 |
(3S)-3-[[(2S)-2-[[(2S,5S,8S,21S)-21-[[2-[[(2S)-5-amino-2-[[2-[2-[2-[(3',6'-dihydroxy-3-oxospiro[2-benzofuran-1,9'-xanthene]-5-yl)carbamothioylamino]ethoxy]ethoxy]acetyl]amino]-5-oxopentanoyl]amino]acetyl]amino]-5-(carboxymethyl)-8,21-dimethyl-2-(2-methylpropyl)-3,6,22-trioxo-1,4,7-triazacyclodocosane-8-carbonyl]amino]-4-methylpentanoyl]amino]-4-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(2-fluorophenyl)-2-methyl-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-4-oxobutanoic acid |
137638518 |
ChemBL |
| YWHAZ |
HGNC:12855 |
P63104 |
(3S)-3-[[(2S)-2-[[(2S,5S,8S,21S)-21-[[2-[[(2S)-5-amino-2-[[2-[2-[2-[(3',6'-dihydroxy-3-oxospiro[2-benzofuran-1,9'-xanthene]-5-yl)carbamothioylamino]ethoxy]ethoxy]acetyl]amino]-5-oxopentanoyl]amino]acetyl]amino]-5-(3-amino-3-oxopropyl)-8,21-dimethyl-2-(2-methylpropyl)-3,6,22-trioxo-1,4,7-triazacyclodocosane-8-carbonyl]amino]-4-methylpentanoyl]amino]-4-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-4-oxobutanoic acid |
137640937 |
ChemBL |
| YWHAZ |
HGNC:12855 |
P63104 |
(3S)-3-[[(2S)-2-[[(2S,5S,8S,21S)-21-[[2-[[(2S)-5-amino-2-[[2-[2-[2-[(3',6'-dihydroxy-3-oxospiro[2-benzofuran-1,9'-xanthene]-5-yl)carbamothioylamino]ethoxy]ethoxy]acetyl]amino]-5-oxopentanoyl]amino]acetyl]amino]-5-(carboxymethyl)-8,21-dimethyl-2-(2-methylpropyl)-3,6,22-trioxo-1,4,7-triazacyclodocosane-8-carbonyl]amino]-4-methylpentanoyl]amino]-4-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-4-oxobutanoic acid |
137647598 |
ChemBL |
| YWHAZ |
HGNC:12855 |
P63104 |
(3S)-3-[[(2S)-2-[[(2S,5S,8S,21S)-21-[[2-[[(2S)-5-amino-2-[[2-[2-[2-[(3',6'-dihydroxy-3-oxospiro[2-benzofuran-1,9'-xanthene]-5-yl)carbamothioylamino]ethoxy]ethoxy]acetyl]amino]-5-oxopentanoyl]amino]acetyl]amino]-5-(carboxymethyl)-8,21-dimethyl-2-(2-methylpropyl)-3,6,22-trioxo-1,4,7-triazacyclodocosane-8-carbonyl]amino]-4-methylpentanoyl]amino]-4-[[(2S)-1-[[(2R)-1-[[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-4-oxobutanoic acid |
137649654 |
ChemBL |
| YWHAZ |
HGNC:12855 |
P63104 |
(3S)-3-[[(2S)-2-[[(2S,5S,8S,21S)-21-[[2-[[(2S)-5-amino-2-[[2-[2-[2-[(3',6'-dihydroxy-3-oxospiro[2-benzofuran-1,9'-xanthene]-5-yl)carbamothioylamino]ethoxy]ethoxy]acetyl]amino]-5-oxopentanoyl]amino]acetyl]amino]-5-(carboxymethyl)-2-(1H-indol-3-ylmethyl)-8,21-dimethyl-3,6,22-trioxo-1,4,7-triazacyclodocosane-8-carbonyl]amino]-4-methylpentanoyl]amino]-4-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-4-oxobutanoic acid |
137652526 |
ChemBL |
| YWHAZ |
HGNC:12855 |
P63104 |
2-[(2S)-3-amino-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S,5S,8S,21S)-21-[[2-[[(2S)-5-amino-2-[[2-[2-[2-[(3',6'-dihydroxy-3-oxospiro[2-benzofuran-1,9'-xanthene]-5-yl)carbamothioylamino]ethoxy]ethoxy]acetyl]amino]-5-oxopentanoyl]amino]acetyl]amino]-5-(carboxymethyl)-8,21-dimethyl-2-(2-methylpropyl)-3,6,22-trioxo-1,4,7-triazacyclodocosane-8-carbonyl]amino]-4-methylpentanoyl]amino]-3-carboxypropanoyl]amino]-4-methylpentanoyl]amino]propanoyl]amino]-3-oxopropyl]propanedioic acid |
137654822 |
ChemBL |
| YWHAZ |
HGNC:12855 |
P63104 |
(3S)-3-[[(2S)-2-[[(2S,5S,8S,21S)-21-[[2-[[(2S)-5-amino-2-[[2-[2-[2-[(3',6'-dihydroxy-3-oxospiro[2-benzofuran-1,9'-xanthene]-5-yl)carbamothioylamino]ethoxy]ethoxy]acetyl]amino]-5-oxopentanoyl]amino]acetyl]amino]-8,21-dimethyl-2-(2-methylpropyl)-5-[3-[(N-nitrocarbamimidoyl)amino]propyl]-3,6,22-trioxo-1,4,7-triazacyclodocosane-8-carbonyl]amino]-4-methylpentanoyl]amino]-4-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-4-oxobutanoic acid |
137659027 |
ChemBL |
| YWHAZ |
HGNC:12855 |
P63104 |
2-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S,5S,8S,21S)-21-[[2-[[(2S)-2-acetamido-5-amino-5-oxopentanoyl]amino]acetyl]amino]-2-(1-adamantyl)-5-(carboxymethyl)-8,21-dimethyl-3,6,22-trioxo-1,4,7-triazacyclodocosane-8-carbonyl]amino]-4-methylpentanoyl]amino]-3-carboxypropanoyl]amino]-4-methylpentanoyl]amino]propanoyl]amino]-3-amino-3-oxopropyl]propanedioic acid |
137659189 |
ChemBL |
| YWHAZ |
HGNC:12855 |
P63104 |
(4aR,6S,7R,8R,8aS)-6-[[(1E,3R,8R,9R,10R,11S,14R)-9-hydroxy-14-methoxy-14-(methoxymethyl)-3,10-dimethyl-6-propan-2-yl-8-tricyclo[9.3.0.03,7]tetradeca-1,6-dienyl]oxy]-2,2-dimethyl-4,4a,6,7,8,8a-hexahydropyrano[3,2-d][1,3]dioxine-7,8-diol |
145974151 |
ChemBL |
| YWHAZ |
HGNC:12855 |
P63104 |
(3S)-4-[[(2S)-1-[(E)-[2-[[(1E,3R,8R,9R,10R,11S,14S)-6-[(2S)-1-acetyloxypropan-2-yl]-8,9-dihydroxy-14-(methoxymethyl)-3,10-dimethyl-4-tricyclo[9.3.0.03,7]tetradeca-1,6-dienyl]oxymethyl]phenyl]methylideneamino]oxy-3-methylbutan-2-yl]amino]-3-[[(2S)-2-[[(2S)-2-[[(2S)-5-amino-2-[[2-[[5-(dimethylamino)naphthalen-1-yl]sulfonylamino]acetyl]amino]-5-oxopentanoyl]amino]-3-hydroxypropanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-4-oxobutanoic acid |
145984749 |
ChemBL |
| YWHAZ |
HGNC:12855 |
P63104 |
(3S)-4-[[(2S)-1-[[(2S)-1-[[(1S)-1-carboxy-2-hydroxyethyl]amino]-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-3-[[(2S,5S,8S,11S,24S)-5-(carboxymethyl)-24-[[2-[[(2S)-2,5-diamino-5-oxopentanoyl]amino]acetyl]amino]-8,11,24-trimethyl-2-(2-methylpropyl)-3,6,9,25-tetraoxo-1,4,7,10-tetrazacyclopentacosane-11-carbonyl]amino]-4-oxobutanoic acid |
145985560 |
ChemBL |
| ZACN |
HGNC:29504 |
Q401N2 |
Tubocurarine |
6000 |
GtoPDB |
| ZACN |
HGNC:29504 |
Q401N2 |
N-(4-tert-butyl-1,3-thiazol-2-yl)-3-fluorobenzamide |
881640 |
GtoPDB |
| MAP3K20 |
HGNC:17797 |
Q9NYL2 |
Sorafenib |
216239 |
DSigDB |
| MAP3K20 |
HGNC:17797 |
Q9NYL2 |
Nilotinib |
644241 |
DSigDB |
| MAP3K20 |
HGNC:17797 |
Q9NYL2 |
Dasatinib |
3062316 |
DSigDB |