GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
ABL1 |
HGNC:76 |
P00519 |
5-(2-aminopyrimidin-4-yl)-2-phenyl-1H-pyrrole-3-carboxamide |
24809764 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
N-(3-(2-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-yl)phenyl)-3-(trifluoromethyl)benzamide |
24822704 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
(E)-methyl 4-(2-(4-bromobenzylthio)-3-(4-fluoro-3-nitrophenyl)acryloyl)benzoate |
24825778 |
TTD |
ABL1 |
HGNC:76 |
P00519 |
3-(2-imidazo[1,2-a]pyrazin-3-ylethynyl)-4-methyl-N-[3-[(4-methylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl]benzamide |
24825841 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
Ponatinib |
24826799 |
BindingDB, TTD |
ABL1 |
HGNC:76 |
P00519 |
3-(Imidazo[1,2-a]pyridin-3-ylethynyl)-4-methyl-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)benzamide |
24827068 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
1-tert-butyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine |
24864305 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
3-(2-aminoquinazolin-6-yl)-4-methyl-1-(4-(oxazol-2-yl)phenyl)pyridin-2(1H)-one |
24879368 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
(S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylamino)-7-(2-methoxyethoxy)quinazolin-6-yl]pyrrolidine-2-carboxamide |
24883334 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
Quizartinib |
24889392 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
4-(2-Chloro-4-fluorophenyl)-8-(2,6-dichlorophenyl)-7-oxido-1,7-naphthyridin-7-ium |
24896769 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
PP121 |
24905142 |
TTD |
ABL1 |
HGNC:76 |
P00519 |
(E)-4-(2-(4-Bromobenzylthio)-3-(4-chloro-3-nitrophenyl)acryloyl)benzoic acid |
24958918 |
BindingDB, TTD |
ABL1 |
HGNC:76 |
P00519 |
(E)-4-(2-(4-Chlorobenzylthio)-3-(4-bromo-3-nitrophenyl)acryloyl)benzoic acid |
24958920 |
TTD |
ABL1 |
HGNC:76 |
P00519 |
(E)-4-(2-(4-Fluorobenzylthio)-3-(4-chloro-3-nitrophenyl)acryloyl)benzoic acid |
24959284 |
TTD |
ABL1 |
HGNC:76 |
P00519 |
(E)-4-(2-(4-Chlorobenzylthio)-3-(4-chloro-3-nitrophenyl)acryloyl)benzoic acid |
24959648 |
BindingDB, TTD |
ABL1 |
HGNC:76 |
P00519 |
(E)-4-(2-(4-Bromobenzylthio)-3-(4-fluoro-3-nitrophenyl)acryloyl)benzoic acid |
24960018 |
TTD |
ABL1 |
HGNC:76 |
P00519 |
(E)-4-(2-(4-Bromobenzylthio)-3-(4-bromo-3-nitrophenyl)acryloyl)benzoic acid |
24960379 |
BindingDB, TTD |
ABL1 |
HGNC:76 |
P00519 |
1H-Pyrazolo[4,3-h]quinazoline-3-carboxamide, 4,5-dihydro-8-[[2-methoxy-5-(4-methyl-1-piperazinyl)phenyl]amino]-1-methyl- |
24993189 |
BindingDB |
ABL1 |
HGNC:76 |
P00519 |
4-[[4-(2-fluoroethyl)piperazin-1-yl]methyl]-N-[4-methyl-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]benzamide |
25017304 |
TTD |