| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MAOB |
[4-Methyl-1,4-dihydro-2H-cyclopenta[b]indol-(3Z)-ylidene]-propyl-amine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
Methyl-carbamic acid 6-chloro-4-methyl-3-[(Z)-methylimino]-1,2,3,4-tetrahydro-cyclopenta[b]indol-7-yl ester |
NA |
395000 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
Methyl-carbamic acid 3-[(Z)-ethylimino]-4-methyl-1,2,3,4-tetrahydro-cyclopenta[b]indol-7-yl ester |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
Methyl-carbamic acid 8-bromo-3-[(Z)-ethylimino]-4-propyl-1,2,3,4-tetrahydro-cyclopenta[b]indol-7-yl ester |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
N-(3-amino-propyl)-N'-(3-benzylamino-propyl)-butane-1,4-diamine |
291000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
1-(1-Methyl-1h-pyrrol-2-yl)-2-phenyl-2-(1-piperidinyl) ethanone |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
2-(Dimethylamino)-1-(1-methyl-1H-pyrrol-2-yl)-2-phenylethan-1-one |
875000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
1-(1-Methyl-1h-pyrrol-2-yl)-2-phenyl-2-(1-pyrrolidinyl) ethanone |
600000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
8-Methoxy-4-methyl-7-(2''-oxocyclopentyloxy)coumarin |
NA |
856000 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
trans-2-Fluoro-2-(3,4-dimethoxyphenyl)cyclopropylamine |
NA |
230000 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
cis-2-Fluoro-2-(3,4-dimethoxyphenyl)cyclopropylamine |
NA |
470000 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
CID 44607264 |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
2-Methyl-9-[9-(2-methyl-1,2,3,4-tetrahydro-beta-carboline-9-yl)nonyl]-1,2,3,4-tetrahydro-beta-carboline |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
9-[9-(beta-Carboline-9-yl)nonyl]-beta-carboline |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
benzyl N-[1-[4-(2-aminocyclopropyl)anilino]-1-oxo-3-phenylpropan-2-yl]carbamate |
133000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
4-Benzyl-1-phenyl-[1,2,4]triazolo[4,3-a]quinoxaline |
NA |
980000 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
Phenyl-(1-phenyl-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl)methanone |
NA |
240000 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
[1-(2-Chlorophenyl)-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl]-phenylmethanone |
NA |
380000 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
[1-[4-(Dimethylamino)phenyl]-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl]-phenylmethanone |
NA |
7300000 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
[1-(4-Nitrophenyl)-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl]-phenylmethanone |
NA |
230000 |
NA |
NA |
NA |
NA |
TTD |