| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MERTK |
US11104676, Example 141 |
NA |
178100 |
NA |
NA |
NA |
NA |
BindingDB |
| MERTK |
US11104676, Example 93 |
NA |
259600 |
NA |
NA |
NA |
NA |
BindingDB |
| MERTK |
US11104676, Example 95 |
NA |
176500 |
NA |
NA |
NA |
NA |
BindingDB |
| MET |
1-N'-[3-fluoro-4-[(2-oxo-1,3-dihydroimidazo[4,5-b]pyridin-7-yl)oxy]phenyl]-1-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide |
NA |
209000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MET |
1-N-(4-fluorophenyl)-1-N'-[3-fluoro-4-(1,3,8-triazatricyclo[7.4.0.02,7]trideca-2,4,6,8-tetraen-6-yloxy)phenyl]cyclopropane-1,1-dicarboxamide |
NA |
260000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MET |
2-[(3-Pyridin-4-yl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)amino]benzoic acid |
NA |
106900 |
NA |
NA |
NA |
NA |
BindingDB |
| MET |
3,3'-Methylenebis(4,7,8-trihydroxy-2h-chromen-2-one) |
NA |
151000 |
NA |
NA |
NA |
NA |
BindingDB |
| MET |
1'-methyl-6-[3-(quinolin-6-ylmethyl)triazolo[4,5-d]pyrimidin-5-yl]spiro[1H-indole-3,4'-piperidine]-2-one |
NA |
1200000 |
NA |
NA |
NA |
NA |
BindingDB |
| MET |
1'-methyl-6-[9-(quinolin-6-ylmethyl)purin-2-yl]spiro[1H-indole-3,4'-piperidine]-2-one |
NA |
1400000 |
NA |
NA |
NA |
NA |
BindingDB |
| MET |
1'-methyl-5-[3-(quinolin-6-ylmethyl)triazolo[4,5-d]pyrimidin-5-yl]spiro[1H-indole-3,4'-piperidine]-2-one |
NA |
140000 |
NA |
NA |
NA |
NA |
BindingDB |
| MET |
1'-methyl-5-[9-(quinolin-6-ylmethyl)purin-2-yl]spiro[1H-indole-3,4'-piperidine]-2-one |
NA |
1100000 |
NA |
NA |
NA |
NA |
BindingDB |
| MET |
6-(2,9-Diazaspiro[5.5]undecan-9-Yl)-9h-Purine |
NA |
183000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MET |
2-cyano-N-(2,5-dibromophenyl)-3-oxobutanamide |
NA |
215000 |
NA |
NA |
NA |
NA |
BindingDB |
| MET |
[4-Amino-2-[[4-(4-methyl-1-piperazinyl)phenyl]amino]-5-thiazolyl](2,3-dihydro-1,4-benzodioxin-6-yl)methanone |
NA |
20000000 |
NA |
NA |
NA |
NA |
TTD |
| MET |
[4-Amino-2-[[4-[4-(1-methylethyl)-1-piperazinyl]phenyl]amino]-5-thiazolyl](3-methoxyphenyl)methanone |
NA |
20000000 |
NA |
NA |
NA |
NA |
TTD |
| METAP1 |
(1-Amino-2-cyclohexylethyl)phosphonic acid |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| METAP1 |
2-(8-Hydroxyquinolin-2-yl)-3-phenyl-1,3-thiazolidin-4-one |
NA |
116100 |
NA |
NA |
NA |
NA |
BindingDB |
| METAP1 |
3-(3-Bromophenyl)-2-(8-hydroxyquinolin-2-yl)-1,3-thiazolidin-4-one |
NA |
112700 |
NA |
NA |
NA |
NA |
BindingDB |
| METAP1 |
3-(4-Bromophenyl)-2-(8-hydroxyquinolin-2-yl)-1,3-thiazolidin-4-one |
NA |
104200 |
NA |
NA |
NA |
NA |
BindingDB |
| METAP1 |
2-(8-Hydroxyquinolin-2-yl)-3-(4-methoxyphenyl)-1,3-thiazolidin-4-one |
NA |
104700 |
NA |
NA |
NA |
NA |
BindingDB |