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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
MKNK2 4-(4-Fluoro-2-propan-2-yloxyanilino)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide NA 219000 NA NA NA NA BindingDB
MKNK2 4-(4-fluoro-2-propan-2-yloxyanilino)-N-(3-methoxypropyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide NA 328000 NA NA NA NA BindingDB
MKNK2 4-(6-Methoxypyridin-3-yl)benzamide NA 108000 NA NA NA NA BindingDB|ChEMBL|TTD
MKNK2 Piperazin-1-yl-(4-pyridin-3-ylphenyl)methanone NA 171000 NA NA NA NA BindingDB|ChEMBL|TTD
MKNK2 N-methyl-4-pyridin-3-ylbenzamide NA 184000 NA NA NA NA BindingDB|ChEMBL|TTD
MKNK2 2-methoxy-4-(1H-pyrazol-4-yl)-N-(2,3,4,5-tetrahydro-1H-3-benzazepin-7-yl)benzamide NA 760000 NA NA NA NA BindingDB|TTD
MLKL Mlkl-IN-1 NA NA 215000 NA NA NA ChEMBL
MLKL (~{S})-1~{H}-benzimidazol-2-yl-(4-propan-2-ylphenyl)methanol NA NA 1807000 NA NA NA ChEMBL
MLKL (S)-1H-benzimidazol-2-yl-(4-methylphenyl)methanol NA NA 3005000 NA NA NA ChEMBL
MLKL 2-[(S)-methoxy-(4-methylphenyl)methyl]-1H-benzimidazole NA NA 821000 NA NA NA ChEMBL
MLKL 2-[(S)-methoxy(naphthalen-2-yl)methyl]-3H-benzimidazole-5-carboxylic acid NA NA 352000 NA NA NA ChEMBL
MLLT3 (2S)-2-[[(2S)-6-amino-2-[[2-[[2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-5-amino-2-[[(2S)-6-amino-2-[[(2S,3R)-2-amino-3-hydroxybutanoyl]amino]hexanoyl]amino]-5-oxopentanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-6-(3-methylbut-2-enoylamino)hexanoyl]amino]-3-hydroxypropanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]acetyl]amino]hexanoyl]amino]propanoic acid NA NA 159000 NA NA NA BindingDB
MLNR Imipenem NA NA NA NA NA 300000 PubChem
MLNR Cefazolin NA NA NA NA NA 300000 PubChem
MLNR Meropenem NA NA NA NA NA 300000 PubChem
MLNR Cefepime NA NA NA NA NA 300000 PubChem
MLNR Ceftazidime NA NA NA NA NA 300000 PubChem
MLNR Aztreonam NA NA NA NA NA 400000 PubChem
MLNR Carumonam NA NA NA NA NA 500000 PubChem
MLNR Doripenem NA NA NA NA NA 300000 PubChem