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Drugs And Genes
Negative Drug Target Genes
Gene
Drug
GENE_SYMBOL
DRUG_NAME
Ki (nM)
IC50 (nM)
Kd (nM)
EC50 (nM)
Potency (nM)
AC50 (nM)
Datasource
MMP2
2-Cinnamamido-N1-hydroxy-N4-pentylsuccinamide
NA
196500
NA
NA
NA
NA
TTD
MMP2
ethyl 5-{1-methyl-3-[(pyridin-4-ylmethyl)carbamoyl]-1H-pyrazol-5-yl}-1H-indole-2-carboxylate
NA
500000
NA
NA
NA
NA
TTD
MMP2
N'-[2-(3-methyl-2-oxo-quinoxalin-1-yl)acetyl]-2-phenyl-acetohydrazide
NA
159390
NA
NA
NA
NA
TTD
MMP2
N'-[2-(3-methyl-2-oxo-quinoxalin-1-yl)acetyl]benzohydrazide
NA
187410
NA
NA
NA
NA
TTD
MMP2
4-(3-Chlorophenylamino)-2-cinnamamido-4-oxobutanoic acid
NA
1000000
NA
NA
NA
NA
TTD
MMP2
N4-(2-Chlorophenyl)-2-cinnamamido-N1-hydroxysuccinamide
NA
1000000
NA
NA
NA
NA
TTD
MMP2
N4-(3-Chlorophenyl)-2-cinnamamido-N1-hydroxysuccinamide
NA
1000000
NA
NA
NA
NA
TTD
MMP2
2-Cinnamamido-4-(isopropylamino)-4-oxobutanoic acid
NA
1000000
NA
NA
NA
NA
TTD
MMP2
4-(Butylamino)-2-cinnamamido-4-oxobutanoic acid
NA
594300
NA
NA
NA
NA
TTD
MMP2
4-(Benzylamino)-2-cinnamamido-4-oxobutanoic acid
NA
999000
NA
NA
NA
NA
TTD
MMP2
N4-Benzyl-2-cinnamamido-N1-hydroxysuccinamide
NA
447200
NA
NA
NA
NA
TTD
MMP2
2-Cinnamamido-4-oxo-4-(pentylamino)butanoic acid
NA
1000000
NA
NA
NA
NA
TTD
MMP2
2-Cinnamamido-4-(hexylamino)-4-oxobutanoic acid
NA
1000000
NA
NA
NA
NA
TTD
MMP2
2-Cinnamamido-4-oxo-4-(phenylamino)butanoic acid
NA
1000000
NA
NA
NA
NA
TTD
MMP2
2-Cinnamamido-N1-hydroxy-N4-phenylsuccinamide
NA
324400
NA
NA
NA
NA
TTD
MMP2
2-Cinnamamido-N1-hydroxy-N4-(3-nitrophenyl)succinamide
NA
1000000
NA
NA
NA
NA
TTD
MMP2
2-Cinnamamido-4-(3-nitrophenylamino)-4-oxobutanoic acid
NA
1000000
NA
NA
NA
NA
TTD
MMP2
2-Cinnamamido-4-(4-nitrophenylamino)-4-oxobutanoic acid
NA
1000000
NA
NA
NA
NA
TTD
MMP2
2-Cinnamamido-4-(octylamino)-4-oxobutanoic acid
NA
1000000
NA
NA
NA
NA
TTD
MMP2
2-Cinnamamido-4-(dodecylamino)-4-oxobutanoic acid
NA
176500
NA
NA
NA
NA
TTD
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