| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| NCK1 |
2-Aminoquinoline |
NA |
NA |
NA |
150000 |
NA |
NA |
BindingDB|TTD |
| NCOA2 |
2-(4-((4-Methylpiperidin-1-yl)sulfonyl)benzamido)thiophene-3-carboxamide |
NA |
NA |
NA |
145500 |
NA |
NA |
BindingDB |
| NCOR1 |
N-(2-Amino-5-fluorophenyl)-4-[[[1-oxo-3-(3-pyridinyl)-2-propen-1-yl]amino]methyl]benzamide |
NA |
180000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| NCSTN |
N-[(3,4-dichlorophenyl)methyl]-N-propan-2-ylnaphthalene-2-carboxamide |
NA |
135000 |
NA |
NA |
NA |
NA |
TTD |
| NCSTN |
9-octyl-2-(2H-tetrazol-5-ylmethoxy)carbazole |
NA |
102000 |
NA |
NA |
NA |
NA |
TTD |
| NCSTN |
2-(9-Octylcarbazol-2-yl)oxyacetamide |
NA |
104000 |
NA |
NA |
NA |
NA |
TTD |
| NCSTN |
2-(9-Octylcarbazol-2-yl)oxyacetonitrile |
NA |
105000 |
NA |
NA |
NA |
NA |
TTD |
| NCSTN |
4-[4-[(Z)-(5-chloro-2-oxo-1H-indol-3-ylidene)methyl]-2-methoxyphenoxy]butanenitrile |
NA |
160000 |
NA |
NA |
NA |
NA |
TTD |
| NCSTN |
Tarenflurbil |
NA |
307000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| NEK2 |
N-methyl-4-[7-(4-methylpiperazin-1-yl)imidazo[1,2-a]pyridin-3-yl]-2-[1-[2-(trifluoromethyl)phenyl]ethoxy]benzamide |
NA |
197000 |
NA |
NA |
NA |
NA |
TTD |
| NEK2 |
4-(7-Chloroimidazo[1,2-a]pyridin-3-yl)-2-[[2-(trifluoromethyl)phenyl]methoxy]benzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| NEU1 |
(2R,3R,4S)-3-acetamido-4-azido-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acid |
NA |
360000 |
NA |
NA |
NA |
NA |
BindingDB |
| NEU1 |
(2R,3R,4S)-3-acetamido-2-[(1R,2R)-3-[4-(4-carboxyphenyl)triazol-1-yl]-1,2-dihydroxypropyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acid |
NA |
240000 |
NA |
NA |
NA |
NA |
BindingDB |
| NEU1 |
(2R,3R,4S)-3-acetamido-2-[(1R,2R)-1,2-dihydroxy-3-[4-[4-(trifluoromethyl)phenyl]triazol-1-yl]propyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acid |
NA |
140000 |
NA |
NA |
NA |
NA |
BindingDB |
| NEU1 |
(2R,3R,4S)-3-acetamido-2-[(1R,2R)-3-[4-[4-(dimethylamino)phenyl]triazol-1-yl]-1,2-dihydroxypropyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acid |
NA |
190000 |
NA |
NA |
NA |
NA |
BindingDB |
| NEU1 |
(2R,3R,4S)-3-(5-aminopentanoylamino)-4-hydroxy-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acid |
NA |
480000 |
NA |
NA |
NA |
NA |
BindingDB |
| NEU1 |
(2R,3R,4S)-3-acetamido-2-[(1R,2R)-3-[5-[(4-acetamidobenzoyl)amino]pentanoylamino]-1,2-dihydroxypropyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acid |
NA |
240000 |
NA |
NA |
NA |
NA |
BindingDB |
| NEU1 |
(2R,3R,4S)-3-[[2-[4-[4-(dimethylamino)phenyl]triazol-1-yl]acetyl]amino]-4-hydroxy-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acid |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB |
| NEU1 |
(2R,3R,4S)-3-acetamido-2-((1R,2R)-3-azido-1,2-dihydroxypropyl)-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylate |
NA |
620000 |
NA |
NA |
NA |
NA |
BindingDB |
| NEU1 |
Peramivir |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem |