| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RAPGEF3 |
(1E)-1-[amino-(4-chloroanilino)methylidene]-2-propan-2-ylguanidine;hydrochloride |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Erythromycin |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Agaricic Acid |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Hydroxychloroquine Sulfate |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Minodronic Acid |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Etonitazene |
NA |
NA |
NA |
NA |
281838 |
NA |
PubChem |
| RAPGEF3 |
Amaranth |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Lithium Citrate |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Tilarginine Acetate |
NA |
NA |
NA |
NA |
112202|125892 |
NA |
PubChem |
| RAPGEF3 |
Clozapine |
NA |
NA |
NA |
NA |
125892|112202 |
NA |
PubChem |
| RAPGEF3 |
Olanzapine |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
8-Hydroxyguanine |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Calcium (4-(((2-amino-5-formyl-4-oxo-1,4,5,6,7,8-hexahydropteridin-6-yl)methyl)amino)benzoyl)glutamate |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
[(7S,11S,12R,13S,14R,15R,16R,17S,18S,19Z,21Z)-2,15,17,27,29-pentahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-26-[(E)-(4-methylpiperazin-1-yl)iminomethyl]-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,25,27-octaen-13-yl] acetate |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
[(7S,11S,12R,13S,14R,15R,16R,17S,18S,19Z,21Z)-26-[(E)-(4-cyclopentylpiperazin-1-yl)iminomethyl]-2,15,17,27,29-pentahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,25,27-octaen-13-yl] acetate |
NA |
NA |
NA |
NA |
125892|112202 |
NA |
PubChem |
| RAPGEF3 |
Estradiol Valerate |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Bunamidine Hydrochloride |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Methadone Hydrochloride |
NA |
NA |
NA |
NA |
223872 |
NA |
PubChem |
| RAPGEF3 |
Methdilazine Hydrochloride |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Amylmetacresol |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |