| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RAPGEF3 |
Flunarizine Hydrochloride |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
cyclosporin A |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Phenoxybenzamine Hydrochloride |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Cyproterone |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Estropipate |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Phytonadione |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
(2S)-2-[(2S,4R,5R,6R)-4-[(2S,4R,5R,6R)-4-[(2S,4S,5R,6R)-4,5-dihydroxy-4,6-dimethyloxan-2-yl]oxy-5-hydroxy-6-methyloxan-2-yl]oxy-5-hydroxy-6-methyloxan-2-yl]oxy-3-[(1S,3S,4R)-3,4-dihydroxy-1-methoxy-2-oxopentyl]-6-[(2S,4R,5S,6R)-4-[(2S,4R,5S,6R)-4,5-dihydroxy-6-methyloxan-2-yl]oxy-5-hydroxy-6-methyloxan-2-yl]oxy-8,9-dihydroxy-7-methyl-3,4-dihydro-2H-anthracen-1-one |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Acipimox |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Vorinostat |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Clobetasol |
NA |
NA |
NA |
NA |
112202|125892 |
NA |
PubChem |
| RAPGEF3 |
Nalbuphine |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Stiripentol |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Andrographolide |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Lovastatin |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Sulfamethizole |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Sulfinpyrazone |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Methoprene |
NA |
NA |
NA |
NA |
112202|125892 |
NA |
PubChem |
| RAPGEF3 |
Gatifloxacin |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Vinblastine Sulfate |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
cis-4-[3-[4-(1,1-Dimethylpropyl)phenyl]-2-methylpropyl]-2,6-dimethylmorpholine |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |