| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RAPGEF3 |
Chlorobutanol |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Ethinyl Estradiol |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Aminopyrine |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Promethazine Hydrochloride |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
(4S)-4-[[(2S)-2-[[(4R)-2-[(1R,2R)-1-amino-2-methylbutyl]-4,5-dihydro-1,3-thiazole-4-carbonyl]amino]-4-methylpentanoyl]amino]-5-[[(2R,3S)-1-[[(3R,6R,9R,12R,15R,18R,21R)-3-(2-amino-2-oxoethyl)-18-(3-aminopropyl)-12-benzyl-15-[(2R)-butan-2-yl]-6-(carboxymethyl)-9-(1H-imidazol-5-ylmethyl)-2,5,8,11,14,17,20-heptaoxo-1,4,7,10,13,16,19-heptazacyclopentacos-21-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-5-oxopentanoic acid |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
acetic acid;cobalt;[(2R,3S,4R,5S)-5-(5,6-dimethylbenzimidazol-1-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] 1-[3-[(1R,2R,3R,5Z,7S,10Z,12S,13S,15Z,17S,18S,19R)-2,13,18-tris(2-amino-2-oxoethyl)-7,12,17-tris(3-amino-3-oxopropyl)-3,5,8,8,13,15,18,19-octamethyl-2,7,12,17-tetrahydro-1H-corrin-24-id-3-yl]propanoylamino]propan-2-yl hydrogen phosphate |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Cephalothin |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Uridine |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Uridine Monophosphate |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Phenylethyl Alcohol |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Topotecan Hydrochloride |
NA |
NA |
NA |
NA |
112202|125892 |
NA |
PubChem |
| RAPGEF3 |
Temoporfin |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Ziprasidone |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Saquinavir Mesylate |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Adenosine |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
1-(-2-Phenethyl)-4-phenyl-4-acetoxypiperidine |
NA |
NA |
NA |
NA |
199526 |
NA |
PubChem |
| RAPGEF3 |
Tolfenamic acid |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Phenelzine Sulfate |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Carbaryl |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Cobaltous sulfate heptahydrate |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |