| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RAPGEF3 |
Diphacinone |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Anthraquinone |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Isopimpinellin |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Trimethobenzamide Hydrochloride |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Clomipramine Hydrochloride |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Econazole Nitrate |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Lomefloxacin Hydrochloride |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Lonazolac |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Isosorbide Dinitrate |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
(1S,2R,3R,6R,7S,8S,9R,10R,12R,13S,15R,17S)-9-{[(2S,3R,4S,6R)-4-(dimethylamino)-3-hydroxy-6-methyloxan-2-yl]oxy}-3-ethyl-2,10-dihydroxy-7-{[(2R,4R,5S,6S)-5-hydroxy-4-methoxy-4,6-dimethyloxan-2-yl]oxy}-15-[(2-methoxyethoxy)methyl]-2,6,8,10,12,17-hexamethyl-4,16-dioxa-14-azabicyclo[11.3.1]heptadecan-5-one |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Itasetron |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Temsirolimus |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
2-Mercaptobenzothiazole |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Chlorothymol |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
D-Serine |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Nefiracetam |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Enrofloxacin |
NA |
NA |
NA |
NA |
125892|112202 |
NA |
PubChem |
| RAPGEF3 |
Midomafetamine hydrochloride |
NA |
NA |
NA |
NA |
316228 |
NA |
PubChem |
| RAPGEF3 |
Danofloxacin |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF3 |
Masoprocol |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |