| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RAPGEF3 |
trans-Thiothixene |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Nandrolone Decanoate |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Methysergide |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Curcumin |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Ergotamine Tartrate |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Alvocidib Hydrochloride |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Pentachlorophenol |
NA |
NA |
NA |
NA |
112202|125892 |
NA |
PubChem |
| RAPGEF3 |
Sorbitan Monooleate |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF3 |
Tocofersolan |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF4 |
Flavone |
NA |
NA |
NA |
NA |
141254 |
NA |
PubChem |
| RAPGEF4 |
2,4,6-trimethyl-N-[3-[2-(2,4,6-trimethylphenyl)ethynyl]phenyl]aniline |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| RAPGEF4 |
Amaranth |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF4 |
Allopurinol |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF4 |
[(7S,11S,12R,13S,14R,15R,16R,17S,18S,19Z,21Z)-2,15,17,27,29-pentahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-26-[(E)-(4-methylpiperazin-1-yl)iminomethyl]-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,25,27-octaen-13-yl] acetate |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF4 |
2-[(5-cyano-4-cyclohexyl-6-oxo-1H-pyrimidin-2-yl)sulfanyl]-N-(4-methylphenyl)acetamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| RAPGEF4 |
2-[(5-cyano-4-cyclohexyl-6-oxo-1H-pyrimidin-2-yl)sulfanyl]acetic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| RAPGEF4 |
2-(2,5-Dimethyl-Benzylsulfanyl)-4-(1-Methyl-Piperidin-4-Yl)-6-Oxo-1,6-Dihydro-Pyrimidine-5-Carbonitrile |
NA |
127000 |
NA |
NA |
NA |
NA |
TTD |
| RAPGEF4 |
4-Cyclohexyl-6-Oxo-2-Phenylamino-1,6-Dihydro-Pyrimidine-5-Carbonitrile |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| RAPGEF4 |
2-(4-Chloro-Phenylamino)-4-Cyclohexyl-6-Oxo-1,6-Dihydro-Pyrimidine-5-Carbonitrile |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| RAPGEF4 |
2-[(5-cyano-4-cyclohexyl-6-oxo-1H-pyrimidin-2-yl)sulfanyl]-N-(2,4,6-trimethylphenyl)acetamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |