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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SLC1A1 (1R,2S)-1-[(2S)-2-amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acid NA 300000 NA NA NA NA TTD
SLC1A1 (1S,2S)-1-[(2S)-2-amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acid NA 300000 NA NA NA NA TTD
SLC1A1 (1R,2R)-1-[(2S)-2-amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acid NA 300000 NA NA NA NA TTD
SLC1A1 (1S,2R)-1-[(2S)-2-amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acid NA 300000 NA NA NA NA TTD
SLC1A1 2-Amino-3-(2,5-dihydro-5-oxo-4-isoxazolyl)propanoic acid NA 1000000 NA NA NA NA TTD
SLC1A1 (2S,3R)-2-amino-3-(benzenesulfonamido)butanedioic acid NA 300000|316228 NA NA NA NA BindingDB|TTD
SLC1A1 (2S)-2-amino-3-(phenoxycarbonylamino)butanedioic acid NA 300000|316228 NA NA NA NA BindingDB|TTD
SLC1A1 (2S)-2-amino-3-[(4-tert-butylphenyl)sulfonylamino]butanedioic acid NA 300000|316228 NA NA NA NA BindingDB|TTD
SLC1A1 (2S)-2-amino-3-[[3-(trifluoromethyl)phenyl]sulfonylamino]butanedioic acid NA 150000|158489 NA NA NA NA BindingDB|TTD
SLC1A1 (2S)-2-amino-3-(4-phenyltriazol-1-yl)butanedioic acid NA 1000000 NA NA NA NA TTD
SLC1A1 (2S)-2-amino-3-benzamidobutanedioic acid NA 1000000 NA NA NA NA BindingDB|TTD
SLC1A1 (2S)-2-amino-3-[(2,3,4,5,6-pentafluorophenyl)sulfonylamino]butanedioic acid NA 150000|158489 NA NA NA NA BindingDB|TTD
SLC1A1 (2S)-2-amino-3-[(3-carboxyphenyl)sulfonylamino]butanedioic acid NA 300000 NA NA NA NA TTD
SLC1A1 (2S)-2-amino-3-[(2,6-dichlorophenyl)sulfonylamino]butanedioic acid NA 300000|316228 NA NA NA NA BindingDB|TTD
SLC1A1 (2S)-2-amino-3-[benzenesulfonyl(methyl)amino]butanedioic acid NA 300000 NA NA NA NA TTD
SLC1A1 (2S)-2-amino-3-[(4-methylsulfonylphenyl)sulfonylamino]butanedioic acid NA 300000|316228 NA NA NA NA BindingDB|TTD
SLC1A1 (2S,4R)-4-(2-carboxyphenoxy)pyrrolidine-2-carboxylic acid;hydrochloride NA 1000000 NA NA NA NA TTD
SLC1A1 (2S,4S)-4-(2-carboxyphenoxy)pyrrolidine-2-carboxylic acid;hydrochloride NA 1000000 NA NA NA NA TTD
SLC1A1 4-chloro-3-[5-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]thiophen-2-yl]benzoic acid NA 300000 NA NA NA NA TTD
SLC1A1 4-chloro-3-[4-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]phenyl]benzoic acid NA 300000 NA NA NA NA TTD