| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| TYRO3 |
US11104676, Example 153 |
NA |
333300 |
NA |
NA |
NA |
NA |
BindingDB |
| TYRO3 |
US11104676, Example 157 |
NA |
118300 |
NA |
NA |
NA |
NA |
BindingDB |
| TYRO3 |
US11104676, Example 158 |
NA |
104000 |
NA |
NA |
NA |
NA |
BindingDB |
| TYRO3 |
US11104676, Example 159 |
NA |
420200 |
NA |
NA |
NA |
NA |
BindingDB |
| TYRO3 |
US11104676, Example 180 |
NA |
140000 |
NA |
NA |
NA |
NA |
BindingDB |
| UBA3 |
Candesartan Cilexetil |
NA |
NA |
195000 |
NA |
NA |
NA |
PubChem |
| UBE2T |
6-(Pyrrolidin-1-yl)nicotinimidamide |
NA |
NA |
550000 |
NA |
NA |
NA |
ChEMBL |
| UBE2T |
1,3-Benzothiazol-2-ylmethylamine |
NA |
NA |
1300000 |
NA |
NA |
NA |
ChEMBL |
| UBLCP1 |
Salicylic Acid |
NA |
66000000 |
NA |
NA |
NA |
NA |
PubChem |
| UCHL1 |
Menadione |
NA |
290000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| UCHL1 |
3-acetyl-2-(4-bromophenyl)-1-[2-(3,4-dichlorophenyl)ethyl]-4-hydroxy-2H-pyrrol-5-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| UCHL1 |
5-(4-butylphenyl)-4-(4-isopropylphenyl)-4H-1,2,4-triazole-3-thiol |
NA |
126000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| UCHL3 |
N-[2-Methoxy-6-(4-methylpiperazin-1-yl)pyridin-3-yl]prop-2-enamide |
NA |
282000 |
NA |
NA |
NA |
NA |
BindingDB |
| UCHL3 |
3-hydroxy-5-(4-methoxyphenyl)-1-(1,3,4-thiadiazol-2-yl)-4-(thiophen-2-ylcarbonyl)-1,5-dihydro-2H-pyrrol-2-one |
NA |
154000 |
NA |
NA |
NA |
NA |
TTD |
| UCHL3 |
2-(4-fluorophenyl)-4-hydroxy-3-(5-methylfuran-2-carbonyl)-1-(pyridin-3-ylmethyl)-2H-pyrrol-5-one |
NA |
123000 |
NA |
NA |
NA |
NA |
TTD |
| UCHL3 |
1-benzyl-3-hydroxy-4-(5-methyl-2-furoyl)-5-(3-pyridinyl)-1,5-dihydro-2H-pyrrol-2-one |
NA |
103000 |
NA |
NA |
NA |
NA |
TTD |
| UCHL3 |
3-acetyl-2-(4-bromophenyl)-1-[2-(3,4-dichlorophenyl)ethyl]-4-hydroxy-2H-pyrrol-5-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| UCHL3 |
5-(4-fluorophenyl)-3-hydroxy-4-[(5-methylfuran-2-yl)carbonyl]-1-(pyridin-3-ylmethyl)-2,5-dihydro-1H-pyrrol-2-one |
NA |
123000 |
NA |
NA |
NA |
NA |
BindingDB |
| UCHL3 |
1-benzyl-3-hydroxy-4-[(5-methylfuran-2-yl)carbonyl]-5-(pyridin-3-yl)-2,5-dihydro-1H-pyrrol-2-one |
NA |
103000 |
NA |
NA |
NA |
NA |
BindingDB |
| UCHL3 |
3-hydroxy-5-(4-methoxyphenyl)-1-(1,3,4-thiadiazol-2-yl)-4-(thiophen-2-ylcarbonyl)-2,5-dihydro-1H-pyrrol-2-one |
NA |
154000 |
NA |
NA |
NA |
NA |
BindingDB |