| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| AKT1 |
N-((S)-1-((S)-1-(benzylamino)-1-oxo-3-phenylpropan-2-ylamino)-3-methyl-1-oxobutan-2-yl)-4-(guanidinomethyl)benzamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| AKT1 |
N-((S)-1-((S)-1-(benzylamino)-1-oxo-3-phenylpropan-2-ylamino)-3-methyl-1-oxobutan-2-yl)-4-(2-guanidinoethyl)benzamide |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| AKT1 |
(2S)-1-[(2S)-2-[(2-acetamidoacetyl)amino]-5-(diaminomethylideneamino)pentanoyl]-N-[(2S)-1-[4-[[(2S)-1-[[(2S)-1-(benzylamino)-1-oxo-3-phenylpropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]carbamoyl]-2-phenylanilino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]pyrrolidine-2-carboxamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| AKT1 |
4-[[(2S)-2-acetamido-5-(diaminomethylideneamino)pentanoyl]amino]-N-[(2S)-1-[[(2S)-1-(benzylamino)-1-oxo-3-phenylpropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]-3-phenylbenzamide |
NA |
288000 |
NA |
NA |
NA |
NA |
TTD |
| AKT1 |
4-[[(2S)-2-acetamido-5-(diaminomethylideneamino)pentanoyl]amino]-N-[(2S)-1-[[(2S)-1-(benzylamino)-1-oxo-3-phenylpropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]-2-phenylbenzamide |
NA |
173000 |
NA |
NA |
NA |
NA |
TTD |
| AKT1 |
Phenylaminoethyl guanidine deriv., 21bb |
NA |
215000 |
NA |
NA |
NA |
NA |
TTD |
| AKT1 |
Phenylaminoethyl guanidine deriv., 21bc |
NA |
152000 |
NA |
NA |
NA |
NA |
TTD |
| AKT1 |
Phenylaminoethyl guanidine deriv., 22aa |
NA |
253000 |
NA |
NA |
NA |
NA |
TTD |
| AKT1 |
Phenylaminoethyl guanidine deriv., 22ba |
NA |
158000 |
NA |
NA |
NA |
NA |
TTD |
| AKT1 |
Indole-aryl scaffold, 36a |
NA |
126000 |
NA |
NA |
NA |
NA |
TTD |
| AKT1 |
Quinazolin-7-yl, 15a |
NA |
112000 |
NA |
NA |
NA |
NA |
TTD |
| AKT1 |
Quinazolin-6-yl, 15b |
NA |
232000 |
NA |
NA |
NA |
NA |
TTD |
| AKT1 |
3-[6-Bromo-3-(4-tert-butylphenyl)imidazo[4,5-b]pyridin-2-yl]pyridin-2-amine |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| AKT1 |
3-(4-Tert-butylphenyl)-2-pyridin-4-ylimidazo[4,5-b]pyridine |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| AKT1 |
3-[6-Bromo-3-[(2-methoxyphenyl)methyl]imidazo[4,5-b]pyridin-2-yl]pyridin-2-amine |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| AKT1 |
3-(4-Tert-butylphenyl)-2-pyridin-3-ylimidazo[4,5-b]pyridine |
NA |
185000 |
NA |
NA |
NA |
NA |
TTD |
| AKT1 |
3-[3-(3-Tert-butylphenyl)imidazo[4,5-b]pyridin-2-yl]pyridin-2-amine |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| AKT1 |
Desmethylxanthohumol |
NA |
143900 |
NA |
NA |
NA |
NA |
TTD |
| AKT1 |
1H-Indazole |
NA |
398107.17 |
NA |
NA |
NA |
NA |
TTD |
| AKT1 |
1H-Pyrrolo(2,3-b)pyridine |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |