| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| F10 |
Mtr-Phe(3-amidino)-NHMe |
190000|190107.83 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
3-[(2S)-2-amino-3-(4-methylsulfonylpiperazin-1-yl)-3-oxopropyl]benzenecarboximidamide |
999000|1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
(2S)-3-(3-carbamimidoylphenyl)-N-methyl-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanamide |
639000|639734.84 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
4-tert-Butoxycarbonylamino-4-{[(4-carbamimidoyl-benzylcarbamoyl)-methyl]-carbamoyl}-butyric acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F10 |
Boc-D-Ser-Gly-NHBn(4-amidino) |
140000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
3-Hydroxy-N-{[4-(N-hydroxycarbamimidoyl)-benzylcarbamoyl]-methyl}-2-phenylmethanesulfonylamino-propionamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F10 |
(1-{[(4-Carbamimidoyl-benzylcarbamoyl)-methyl]-carbamoyl}-2-hydroxy-ethyl)-carbamic acid benzyl ester |
140000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
(2S)-1-[(2R)-2-(benzylsulfonylamino)-3-cyclohexylpropanoyl]-N-(5,6,7,8-tetrahydroquinazolin-6-ylmethyl)pyrrolidine-2-carboxamide |
111000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
1-[5-(Diaminomethyl-amino)-2-(3-methyl-1,2,3,4-tetrahydro-quinoline-8-sulfonylamino)-pentanoyl]-4-methyl-piperidine-2-carboxylic acid |
210000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
N-[(2S)-6-amino-1-[5-[[4-[2-(3,4-dichlorophenyl)ethoxy]phenyl]methyl]-1,2,4-oxadiazol-3-yl]-1-oxohexan-2-yl]-3,4-difluorobenzamide |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F10 |
N-[4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-benzyl]-guanidine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| F10 |
N-{2-[4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-phenyl]-ethyl}-guanidine trifluoro-acetic acid |
NA |
175400 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
N-[4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-phenyl]-guanidine trifluoro-acetic acid |
NA |
129000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
2-[2-[(3-Carbamoylphenyl)carbamoyl]-4-(methylamino)phenyl]-5-(2-methylpropylcarbamoyl)benzoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| F10 |
2-[2-[(3-carbamoylphenyl)carbamoyl]-4-(methylamino)phenyl]-5-[[(1S)-1-carboxy-3-methylbutyl]carbamoyl]benzoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| F10 |
5-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]carbamoyl]-2-[2-[(3-carbamoylphenyl)carbamoyl]-4-(methylamino)phenyl]benzoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| F10 |
(4-Guanidino-benzyl)-carbamic acid benzyl ester |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F10 |
[Amino(phenyl)methylidene]azanium |
110000|165000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| F10 |
3-Amino-N-{3-[(S)-2-[4-(2-amino-ethyl)-piperidin-1-yl]-1-(4-aminomethyl-benzyl)-2-oxo-ethylsulfamoyl]-phenyl}-propionamide |
430000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
methyl (2S)-1-[(2S)-2-[[3-(3-aminopropanoylamino)phenyl]sulfonylamino]-3-(3-carbamimidoylphenyl)propanoyl]piperidine-2-carboxylate |
127000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |