| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| F11 |
sodium;[3-ethoxycarbonyl-2-[(3-ethoxycarbonyl-2-methyl-1H-indol-5-yl)oxymethyl]-1-[(2-methylpropan-2-yl)oxycarbonyl]indol-5-yl] sulfate |
NA |
220000 |
NA |
NA |
NA |
NA |
TTD |
| F11 |
[2-[[6-Methoxy-3-[(2-methylpropan-2-yl)oxycarbonyl]-1-benzofuran-5-yl]oxymethyl]-1,3-benzothiazol-6-yl] sulfate |
NA |
124000 |
NA |
NA |
NA |
NA |
BindingDB |
| F11 |
[2-[(2-benzyl-3-ethoxycarbonyl-6-methoxy-1-benzofuran-5-yl)oxymethyl]-3-ethoxycarbonyl-1H-indol-5-yl] sulfate |
NA |
118000 |
NA |
NA |
NA |
NA |
BindingDB |
| F11 |
[3-ethoxycarbonyl-2-[(3-ethoxycarbonyl-2-methyl-1H-indol-5-yl)oxymethyl]-1-[(2-methylpropan-2-yl)oxycarbonyl]indol-5-yl] sulfate |
NA |
220000 |
NA |
NA |
NA |
NA |
BindingDB |
| F11 |
Pentasodium;[4-[3-[8-[4-[[2-(3,4-disulfonatooxyphenyl)-4-oxo-3,7-disulfonatooxychromen-5-yl]oxymethyl]triazol-1-yl]octyl]-4-oxoquinazolin-2-yl]phenyl] sulfate |
NA |
133000 |
NA |
NA |
NA |
NA |
BindingDB |
| F11 |
N-[(6-amino-2-methylpyridin-3-yl)methyl]-1-[[4-(pyrazol-1-ylmethyl)phenyl]methyl]pyrazole-4-carboxamide |
NA |
106000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F11 |
sodium;[4-(4-oxo-3H-quinazolin-2-yl)phenyl] sulfate |
NA |
NA|375000 |
365000|NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| F11 |
2-(3,4-Dihydroxyphenyl)-5-[[4-[[2-(3,4-dihydroxyphenyl)-3,7-dihydroxy-4-oxochromen-5-yl]oxymethyl]phenyl]methoxy]-3,7-dihydroxychromen-4-one |
NA |
208000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F11 |
Octasodium;[2-(3,4-disulfonatooxyphenyl)-5-[[4-[[2-(3,4-disulfonatooxyphenyl)-4-oxo-3,7-disulfonatooxychromen-5-yl]oxymethyl]phenyl]methoxy]-4-oxo-3-sulfonatooxychromen-7-yl] sulfate |
NA |
180000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F11 |
4-hydroxy-N-[(2S)-1-(methylamino)-1-oxo-3-phenylpropan-2-yl]-2-oxo-1H-quinoline-6-carboxamide |
NA |
NA |
1400000 |
NA |
NA |
NA |
BindingDB |
| F11 |
2-(3-Cyano-4-hydroxyphenyl)-3-hydroxy-5-methylimidazole-4-carboxylic acid |
228000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| F11 |
2-(3-Cyanophenyl)-3-hydroxy-5-methylimidazole-4-carboxylic acid |
120000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| F11 |
Pentasodium;[4-[3-[7-[4-[[2-(3,4-disulfonatooxyphenyl)-4-oxo-3,7-disulfonatooxychromen-5-yl]oxymethyl]triazol-1-yl]heptyl]-4-oxoquinazolin-2-yl]phenyl] sulfate |
NA |
139000 |
NA |
NA |
NA |
NA |
BindingDB |
| F11 |
disodium;[3-[4-oxo-3-[(E)-4-[4-oxo-2-(3-sulfonatooxyphenyl)quinazolin-3-yl]but-2-enyl]quinazolin-2-yl]phenyl] sulfate |
NA |
415000 |
NA |
NA |
NA |
NA |
BindingDB |
| F11 |
Disodium;[3-[4-oxo-3-[[4-[[4-oxo-2-(3-sulfonatooxyphenyl)quinazolin-3-yl]methyl]phenyl]methyl]quinazolin-2-yl]phenyl] sulfate |
NA |
248000 |
NA |
NA |
NA |
NA |
BindingDB |
| F11 |
Disodium;[3-[4-oxo-3-[2-[2-[4-oxo-2-(3-sulfonatooxyphenyl)quinazolin-3-yl]ethoxy]ethyl]quinazolin-2-yl]phenyl] sulfate |
NA |
401000 |
NA |
NA |
NA |
NA |
BindingDB |
| F11 |
Benzamidine |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB |
| F11 |
6-Chloro-2-hydroxyquinoline |
NA |
140000 |
NA |
NA |
NA |
NA |
BindingDB |
| F11 |
(1R,6S,8S,8aS)-6-Amino-6-cyclohex-1-enylmethyl-1-ethyl-8-methoxy-5-oxo-octahydro-indolizine-3-carboxylic acid 4-carbamimidoyl-benzylamide; hydrochloride |
NA |
133000 |
NA |
NA |
NA |
NA |
TTD |
| F11 |
(1R,6S,8S,8aS)-6-Amino-6-benzyl-1-ethyl-8-methoxy-5-oxo-octahydro-indolizine-3-carboxylic acid 4-carbamimidoyl-benzylamide; hydrochloride |
NA |
133000 |
NA |
NA |
NA |
NA |
TTD |