| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| F2 |
[5-[4-[[4-[(E)-N'-methoxycarbonylcarbamimidoyl]phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-(2-piperidin-4-ylethylcarbamoyl)piperazine-1-carboxylate |
561000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
1,4-Di[4-(4-aminomethylhexahydro-1-pyridinylcarboxamidomethyl)hexahydro-1-pyridinylcarbonyloxymethyl]benzene |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
{4-[(4-Aminomethyl-piperidine-1-carbonyl)-amino]-butyl}-carbamic acid 4-{4-[(4-aminomethyl-piperidine-1-carbonyl)-amino]-butylcarbamoyloxymethyl}-benzyl ester |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
[5-[4-[[(4-Carbamimidoylphenyl)sulfonylamino]methyl]piperidine-1-carbonyl]oxycyclooctyl] 4-(2-piperidin-4-ylethylcarbamoyl)piperazine-1-carboxylate |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
5-[(1R,3aS,8bS)-2-oxo-3,3a,4,8b-tetrahydro-1H-indeno[2,1-b]pyrrol-1-yl]pentanimidamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
1-(4-Benzyloxy-benzyl)-pyridinium |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-[3-(3-Benzyl-1H-indol-2-yl)-5-bromo-4-hydroxy-phenyl]-propionic acid |
700000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3,4,5,6-Tetrahydro-2H-[1,4'']bipyridinyl-4-carboxylic acid [2-(3-carbamimidoyl-phenoxy)-ethyl]-amide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
N-[2-(3-Carbamimidoyl-phenoxy)-ethyl]-benzamide |
800000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
5-Bromo-N-(4-guanidino-phenyl)-2-hydroxy-benzamide |
450000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
N-(4-Guanidino-phenyl)-2-hydroxy-5-nitro-benzamide |
315000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
N-(4-Guanidino-phenyl)-2-hydroxy-benzamide |
450000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
2-Hydroxy-biphenyl-3-carboxylic acid (4-carbamimidoyl-phenyl)-amide |
120000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
N-(4-Carbamimidoyl-phenyl)-2-hydroxy-5-nitro-benzamide |
185000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
4-Ethoxy-N-(4-guanidino-phenyl)-2-hydroxy-benzamide |
450000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
N-(4-Guanidino-phenyl)-2-hydroxy-5-methyl-benzamide |
450000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-Hydroxy-4-isopropoxy-anthracene-2-carboxylic acid (4-guanidino-phenyl)-amide |
450000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-Hydroxy-4-isopropoxy-anthracene-2-carboxylic acid (6-guanidino-pyridin-3-yl)-amide |
450000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-Hydroxy-4-methoxy-anthracene-2-carboxylic acid (6-guanidino-pyridin-3-yl)-amide |
195000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
N-(4-Guanidino-phenyl)-2-hydroxy-4-methyl-benzamide |
450000 |
NA |
NA |
NA |
NA |
NA |
TTD |