Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| HDAC6 | 8-[2-[[(5S,5aS,8aR,9R)-9-(4-hydroxy-3,5-dimethoxyphenyl)-8-oxo-5a,6,8a,9-tetrahydro-5H-[2]benzofuro[5,6-f][1,3]benzodioxol-5-yl]amino]phenoxy]-N-hydroxyoctanamide | NA | 217000 | NA | NA | NA | NA | TTD |
| HDAC6 | N-hydroxy-2-[4-[3-[4-(2-hydroxy-3,3-dimethylbutoxy)-3-methylphenyl]pentan-3-yl]-2-methylphenoxy]acetamide | NA | 580000 | NA | NA | NA | NA | BindingDB |
| HDAC6 | 2-(4-Oxo-3,4-dihydroquinazolin-3-yl)acetic acid | NA | 320000 | NA | NA | NA | NA | BindingDB|TTD |
| HDAC6 | 3-(1,3-Benzothiazol-2-yl)propanoic acid | NA | 180000 | NA | NA | NA | NA | BindingDB|TTD |
| HDAC6 | NA | NA | 150000 | NA | NA | NA | BindingDB | |
| HDAC6 | 8-Mercaptoquinoline | NA | 200000 | NA | NA | NA | NA | TTD |
| HDAC6 | Curcumin | NA | 187000 | NA | NA | NA | NA | PubChem |
| HDAC6 | N-(2-Amino-5-fluorophenyl)-4-[[[1-oxo-3-(3-pyridinyl)-2-propen-1-yl]amino]methyl]benzamide | NA | 1000000 | NA | NA | NA | NA | PubChem |
| HDAC6 | NA | NA | 200000 | NA | NA | NA | BindingDB | |
| HDAC7 | Acetylcysteine | NA | 3160000 | NA | NA | NA | NA | PubChem |
| HDAC7 | N-Hydroxy-E-3-(4''-methoxybiphenyl-4-yl)-acrylamide | NA | 210000|213000 | NA | NA | NA | NA | BindingDB|TTD |
| HDAC7 | Chlorogenic Acid | NA | 375000|200000 | NA | NA | NA | NA | PubChem |
| HDAC7 | Butyric Acid | NA|136000 | 300000|NA|2000000 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| HDAC7 | N-hydroxy-4-phenylbutanamide | NA | 150000 | NA | NA | NA | NA | BindingDB|TTD |
| HDAC7 | Valproic Acid | NA|564000 | 2000000|995000|7240000|NA | NA | NA | NA | NA | PubChem|TTD |
| HDAC7 | N-hydroxybutanamide | NA | 1000000 | NA | NA | NA | NA | TTD |
| HDAC7 | Phenylbutyric acid | NA | 2000000 | NA | NA | NA | NA | PubChem|TTD |
| HDAC7 | Sodium Butyrate | NA|365000 | 140000|NA|800000 | NA | NA | NA | NA | PubChem |
| HDAC7 | (1E,4Z,6E)-5-hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-one | NA | 115000 | NA | NA | NA | NA | PubChem |
| HDAC7 | Vorinostat | NA | 105000|110000 | NA | NA | NA | NA | BindingDB|PubChem |