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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
HDAC8 methyl (2S)-2-acetamido-3-(4-phenylmethoxyphenyl)propanoate NA 871500 NA NA NA NA BindingDB|TTD
HDAC8 (2S)-2-[(4-methylbenzoyl)amino]-3-(4-phenylmethoxyphenyl)propanoic acid NA 1000000 NA NA NA NA TTD
HDAC8 (2S)-2-(methanesulfonamido)-3-[4-(2-phenylethoxy)phenyl]propanoic acid NA 102300 NA NA NA NA BindingDB|TTD
HDAC8 methyl (2S)-2-benzamido-3-[4-(2-phenylethoxy)phenyl]propanoate NA 1000000 NA NA NA NA TTD
HDAC8 (2S)-2-[(4-methylbenzoyl)amino]-3-[4-(2-phenylethoxy)phenyl]propanoic acid NA 385600 NA NA NA NA BindingDB|TTD
HDAC8 (2S)-2-acetamido-3-[4-(2-phenylethoxy)phenyl]propanoic acid NA 120900 NA NA NA NA BindingDB|TTD
HDAC8 (2S)-2-[(4-methylphenyl)sulfonylamino]-3-[4-(2-phenylethoxy)phenyl]propanoic acid NA 1000000 NA NA NA NA TTD
HDAC8 methyl (2S)-2-(methanesulfonamido)-3-[4-(2-phenylethoxy)phenyl]propanoate NA 1000000 NA NA NA NA TTD
HDAC8 methyl (2S)-2-[(4-methylphenyl)sulfonylamino]-3-[4-(2-phenylethoxy)phenyl]propanoate NA 961800 NA NA NA NA BindingDB|TTD
HDAC8 (2S)-2-benzamido-3-[4-(2-phenylethoxy)phenyl]propanoic acid NA 253400 NA NA NA NA BindingDB|TTD
HDAC8 Ubenimex NA 1000000 NA NA NA NA PubChem
HDAC8 5-Amino-N-hydroxypentanamide (4) NA 120000 NA NA NA NA BindingDB
HDAC8 Curcumin NA 187000 NA NA NA NA PubChem
HDAC8 N-(2-Amino-5-fluorophenyl)-4-[[[1-oxo-3-(3-pyridinyl)-2-propen-1-yl]amino]methyl]benzamide NA 1000000 NA NA NA NA PubChem
HDAC9 Acetylcysteine NA 3160000 NA NA NA NA PubChem
HDAC9 Chlorogenic Acid NA 375000|200000 NA NA NA NA PubChem
HDAC9 Butyric Acid 136000|NA NA|2000000 NA NA NA NA PubChem|TTD
HDAC9 N-hydroxy-4-phenylbutanamide NA 430000 NA NA NA NA BindingDB|TTD
HDAC9 Valproic Acid 564000|NA NA|995000|7240000|2000000 NA NA NA NA PubChem|TTD
HDAC9 N-hydroxybutanamide NA 2000000 NA NA NA NA TTD